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2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-methyl-N-[3-(pyrrolidin-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
N2,N2,6-trimethyl-N4-[3-(pyrrolidin-1-yl)propyl]pyrimidine-2,4-diamine
8-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2-methyl-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-[2-(benzyloxy)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxy-4-{[(2-methylpropyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-phenylpyrimidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
N,4-dimethyl-5-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(2,2-diphenylethyl)-4-methylazepan-4-ol
(1s,4s)-4-{4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
4-[(5-chlorothiophen-2-yl)methyl]-9-(2-methoxyethyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(oxan-4-yl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-{[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(1R,7S)-N-methyl-4-oxo-3-[2-(piperidin-1-yl)ethyl]-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-[3-(pyridin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-(2-{[3-(pyridin-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
(2S,3S)-2-amino-1-(4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-methylpentan-1-one
N-cyclopropyl-5-(2-methyl-5-propylpyrimidin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-(cyclopropylsulfamoyl)-5-[4-(dimethylcarbamoyl)phenyl]benzoic acid
methyl 2-{5-[1-(3-methylpyrazin-2-yl)piperidin-4-yl]-1H-pyrazol-3-yl}acetate
4-{[1-(5-propyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}pyridine
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-[3-methyl-1-(4-methylphenyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzoic acid
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
(2R,3R,6R)-5-(1,8-naphthyridine-2-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
5-(4-chloro-2-methoxyphenoxymethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(3-methyloxetan-3-yl)methyl]amine
1-[2-methoxy-4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2,2-dimethyl-N-{[1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methyl}propanamide
2-{[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
2-(3-chlorophenyl)-4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
4-{[2-(2-phenylethyl)piperidin-1-yl]sulfonyl}morpholine
N1-(pyridin-3-yl)-N3-(thiolan-3-yl)propane-1,3-diamine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(1S,6R)-9-(1,4-dimethyl-1H-indole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-(2,3-dihydro-1H-inden-2-yl)-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-[4-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
3-(4-methoxy-2-methylbenzoyl)piperidine
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[2-(benzyloxy)ethyl]-2,3-dihydropyridazin-3-one
N-[(1-hydroxycyclohexyl)methyl]-4-propylpyrimidine-5-carboxamide
1-ethyl-N-[(1-phenylcyclopentyl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(2-{1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-{1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]formamido}acetamide
1-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-methoxypropan-2-ol