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N-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-dichlorobenzamide
2-(4-fluorophenoxy)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
1-[1-({3-[hydroxy(phenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}methyl)-3,5-dimethyl-1H-pyrazol-4-yl]ethan-1-one
3-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
1-cyclopropyl-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-2-one
3-(3-hydroxy-3-methylbutyl)-N-[(1R,2S)-2-hydroxycyclohexyl]-N-methylbenzamide
(1S,5R)-3-{[3-(2-aminoethyl)phenyl]methyl}-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-[2-(dimethylamino)phenyl]-1H-pyrazol-1-yl}-N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-(methylsulfanyl)-1H-1,2,4-triazole
N-[2-(1H-pyrazol-1-yl)ethyl]-2-(quinazolin-4-yloxy)acetamide
N4-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-5-methylpyrimidine-2,4-diamine
N-cyclopentyl-3-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-oxopentanamide
N-(2,3-dihydro-1H-inden-1-yl)-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-[2-(3-methoxyphenyl)phenyl]-1-(1H-pyrrole-3-carbonyl)piperidine-4-carboxamide
2-methyl-1-{1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]azetidin-3-yl}piperidine
2-(4-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(5-fluoro-2-methylphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
1-methyl-2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
N-benzyl-3-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-N-methylpropanamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{[1-cyclohexyl-3-(cyclopropylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl]formamido}propanamide
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-(4-fluorophenyl)piperidin-3-amine
(3S,4S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(dimethylamino)pyrrolidin-3-ol
(3E)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pent-3-enamide
N,N-dimethyl-4-(3-methyl-1H-pyrazol-5-yl)-5,6,7,8-tetrahydroquinazolin-2-amine
1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]-3-(thiophen-2-ylmethyl)urea
N,1-bis(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]-1H-1,3-benzodiazole-5-sulfonamide
3-methyl-N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
6-ethyl-4-(7-methoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-dihydropyridin-2-one
2-{5-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2-phenylpropyl)piperidine
4-(1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
(1H-indazol-3-ylmethyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
1-{3-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]phenyl}ethan-1-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-(4-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine
8-(2,3-dihydro-1H-inden-2-yl)-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-fluorophenyl)-N-[(1R)-2-hydroxy-1-phenylethyl]imidazo[1,2-a]pyridine-6-carboxamide
(3R,4S)-4-[4-(3,5-dichloro-4-methylbenzoyl)-1,4-diazepan-1-yl]oxolan-3-ol
N,N,1-trimethyl-4-{[3-(methylsulfanyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
4-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine
3-[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]pyridin-2-ol
ethyl 2-(methylsulfanyl)-4-(quinolin-8-yl)pyrimidine-5-carboxylate
2-{4-[1-(1-methylcyclohexanecarbonyl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
3-[(4-fluorophenyl)methyl]-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]benzoic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[(5-fluoro-2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
(2R,3R)-3-({[1-(dimethylamino)cycloheptyl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol