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[(2,4-dimethoxy-3-methylphenyl)methyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-(2-methoxyethyl)-4-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]pyrrolidin-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-chloro-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-4-propoxybenzamide
1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-(4H-1,2,4-triazol-4-yl)piperidine
2-(dimethylamino)-N-{2-[ethyl(methyl)amino]-2-methylpropyl}-2-(4-fluorophenyl)acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)piperidine-3-carboxamide
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,4-diazepane-1-carbaldehyde
2-[3-(propanamidomethyl)phenyl]benzamide
1-{3-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-(propan-2-yl)acetamide
7-[(3-methylphenyl)methyl]-2-(1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-{[2-(phenylcarbamoyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(2-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
4-{[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)carbamoyl}pyridin-1-ium-1-olate
methyl 2-(5-oxo-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepane-1-carbonyl)benzoate
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
3-[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]-1-(4-benzylpiperidin-1-yl)propan-1-one
3-(2,4-difluorophenyl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(2-aminoethyl)-N-[2-(3-methylthiophen-2-yl)ethyl]quinazolin-4-amine
N-cyclooctyl-4-[2-(3-methoxypropyl)piperidin-1-yl]-4-oxobutanamide
(2S,4S)-4-amino-1-(3-acetamidobenzenesulfonyl)-N-ethylpyrrolidine-2-carboxamide
2-(2-methoxyethyl)-9-[3-(2-methyl-1H-imidazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(cyclohexylmethyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3S,4S)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
N'1-[(4-fluorophenyl)(pyridin-4-yl)methyl]cyclopropane-1,1-dicarboxamide
(3S,4S)-4-cyclopropyl-1-[4-(morpholin-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
2-[2-(1H-imidazol-1-yl)ethyl]-1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(2-methoxyphenyl)benzamide
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-methyl-1H-indazole-3-carboxamide
N-butyl-1-cyclohexyl-3-(cyclopropylmethyl)-N-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazol-4-yl}piperidine
(3S,4R)-1-(9H-purin-6-yl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
3,4-dimethoxy-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}pyridine
1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(1-ethylcyclopropyl)methyl]acetamide
(3S,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-1-(2-methoxyacetyl)-N-methylpiperidine-3-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
N-[2-(1H-imidazol-4-yl)ethyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(1R,5R)-6-(6-fluoro-1H-1,3-benzodiazole-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-{[4-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-1-yl]methyl}phenol
methyl 3-[1-(4-methylpentanoyl)piperidin-4-yl]propanoate
(3S,4S)-4-cyclopropyl-1-(1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
8-chloro-2-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]quinolin-4-ol
2-{4-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]morpholin-3-yl}-N-phenylacetamide