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6-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-methylpyrimidin-4-amine
(3R,4S)-4-cyclopropyl-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-amine
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}butanamide
N-[(2-ethoxypyridin-3-yl)methyl]-2-(1H-imidazol-2-yl)benzamide
4,6-dimethyl-2-oxo-N-(2-phenoxyethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-ethoxy-5-{2-[(quinolin-3-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}benzamide
N-methyl-3-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyridin-2-amine
4-(1H-imidazol-1-ylmethyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-phenyl-1,3,4-oxadiazole
3-[5-(3-methyl-1,2-oxazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-3-methyl-1H-indole-2-carboxamide
2-(2,4-difluorophenoxy)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
2-[5-(methoxymethyl)-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
N-[(1S,2R)-2-aminocyclobutyl]-2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-cyclohexyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(pyridin-2-ylmethyl)acetamide
(1S,5R)-3-{5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3,5-dimethyl-1,2-oxazole-4-sulfonamide
1-{3-[4-(4-fluorophenyl)-4-hydroxypiperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
1-(2-aminoethyl)-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(2,2-dimethylpropyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
(3S,4S)-1-(5-ethylthiophene-3-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[3-(2,4-dimethoxyphenyl)phenyl]-5-methyl-1,3,4-thiadiazole
1-(3,5-dimethylphenyl)-4-(3-methylfuran-2-carbonyl)piperazin-2-one
2-{methyl[(4-methyl-5-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amino}ethan-1-ol
5-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-1,3-thiazol-4-yl]methanol
{[(3S,4R)-1-(4-chloro-2-methylbenzoyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-[2-fluoro-5-({methyl[2-(pyridin-4-yl)ethyl]carbamoyl}amino)phenyl]-2-methylpropanamide
{4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-1,4-oxazepan-6-yl}methanol
N-[1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)piperidin-3-yl]acetamide
5-{[2-(diethylamino)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1,3-dimethyl-2,6-dioxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-N-(pyrimidin-4-ylmethyl)-2,3-dihydro-1H-isoindole-4-carboxamide
3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-phenyl-5-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1H-pyrrole
2,3-dimethyl-6-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-[(3S,4R)-1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(thiophen-3-yl)ethan-1-one
1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-6-(thian-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
3-(2-phenylpropyl)-8-(pyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-3-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]phenol
{5-[(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
1-[4-fluoro-3-(1H-pyrazol-3-yl)phenyl]ethan-1-one
N-(3-chloro-2-propoxyphenyl)-4-(5-methylpyrimidin-4-yl)piperidine-1-carboxamide
(3S,7S)-5-[5-(propan-2-yl)pyrimidin-4-yl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(1-{4-[2-(morpholin-4-ylmethyl)phenyl]phenyl}ethyl)acetamide