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4-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-2-one
1-[4-(2-amino-6-methoxypyrimidin-4-yl)phenyl]ethan-1-one
N-{[5-(2-methylpentyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}methanesulfonamide
1-[6-(2-methoxypyridin-3-yl)pyridin-2-yl]piperazine
N-(2-methoxyethyl)-N,5-dimethyl-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-benzyl-3-ethyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,4-diazepan-5-one
N-[(3R,4S)-1-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-4-propylpyrrolidin-3-yl]acetamide
1-(3-chlorophenyl)-4-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]piperazine
(4aS,8aS)-2-cyclopentanecarbonyl-7-(3-methyl-1,2-oxazole-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
(2S,4S)-N-(adamantan-2-yl)-4-(3-methoxypropanamido)-1-methylpyrrolidine-2-carboxamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[(2-ethoxyphenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
7-(cyclobutylmethyl)-2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[1-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
1-(1-{2-[(prop-2-en-1-yl)amino]benzoyl}-1,2,3,6-tetrahydropyridin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-ethyl-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
7-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-(2-fluoro-5-methylphenyl)-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propanamide
2-(4-methoxy-2-methylphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
{[1-({1-[(5-methylthiophen-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}urea
2-chloro-5-({4-phenyl-5-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-1-yl}methyl)pyridine
3-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
7-chloro-2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-1H-indole
4-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
1-(6-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}pyrimidin-4-yl)piperidin-4-ol
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]ethan-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-4-methylpyridine-3-carboxamide
N,N-dimethyl-5-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
dimethyl({3-[2-(morpholin-4-ylmethyl)phenoxy]propyl})amine
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
2-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-5,8-dimethylquinolin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(oxan-4-yl)piperidin-3-ol
7-(cyclopropylmethyl)-2-(5-phenoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(8R,9aS)-8-hydroxy-2-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-[(3-methoxyphenyl)methyl]-8-methyl-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 5-[3-(methylsulfanyl)propanoyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-N-ethyl-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
1-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
methyl 3-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methoxy}pyridine-2-carboxylate
3-({3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[1-(1-benzyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)ethyl]methanesulfonamide
N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-3-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-cyclopentyl-5-(2-ethylpiperidine-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-acetyl-1H-1,3-benzodiazol-1-yl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide