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2-(3-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-amine
1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
3-methyl-5-({4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}methyl)-4H-1,2,4-triazole
2-[3-methyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]ethan-1-amine
3-benzyl-8-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(5-chloropyridin-2-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(2,4-difluorophenyl)ethyl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
ethyl 1-{[7-fluoro-2-oxo-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-3-yl]methyl}piperidine-4-carboxylate
3-(4-chloro-2,6-dimethylphenyl)-1-methyl-1-[2-(2-oxopiperidin-1-yl)ethyl]urea
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
1-[2-(piperidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
4-(4-fluorophenyl)-N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-4-oxobutanamide
(4aR,7aS)-1-acetyl-4-(4-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]propanamide
3-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(pyridin-3-yl)propanamide
1-(1-{1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)cyclopentan-1-ol
1,4-dimethyl-9-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1,4,9-triazaspiro[5.5]undecane
2-(dimethylamino)-2-(2-fluorophenyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}acetamide
N3-cyclopentyl-N5-(2,2-dimethyloxan-4-yl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[1-(2-propoxyethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
1-ethyl-N-methyl-3-(2-methylpropyl)-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
2-[2-(4-fluorophenyl)piperidin-1-yl]-1-(piperazin-1-yl)ethan-1-one
(2S,4S)-4-amino-1-(3-{[(4-fluorophenyl)methyl]amino}benzoyl)-N-methylpyrrolidine-2-carboxamide
1-(1-{[1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-[4-({[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(5S,9aS,9bS)-5-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(2-chlorophenoxy)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
ethyl 3-[(4-fluorophenyl)methyl]-1-(quinoline-3-carbonyl)piperidine-3-carboxylate
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}imidazo[1,2-b]pyridazine-3-carboxamide
N-methyl-5-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
(2E)-1-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]-4-methylpent-2-en-1-one
2-(5-fluoro-2-methoxyphenyl)-2-[(furan-3-ylmethyl)(methyl)amino]acetic acid
3-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-3-ylmethyl)benzamide
1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[6-(cyclopropylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl](methyl)amino}methyl)-1-ethylpyrrolidin-2-one
8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[4.5]decan-3-one
3-({[(1-ethylcyclopropyl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-methyl-6-(pyridin-4-yl)pyrimidin-2-amine
2-(4-ethylpiperazin-1-yl)-N-[2-(oxan-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
4-(2-phenoxyethyl)-1-(1-phenylcyclopropanecarbonyl)-1,4-diazepan-5-one
9-[2-(2-ethoxyphenyl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]-N,6-dimethylpyrimidin-4-amine
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-3-fluoro-N-(2-methoxyethyl)benzamide
2-(methylsulfanyl)-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one