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N-[(3S,4R)-1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
8-(3-fluoropyridin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}benzamide
2-[(2-methoxypyridin-3-yl)methyl]-2-azaspiro[4.5]decan-3-one
1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidin-4-amine
2-methoxy-3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazine
2-methoxy-6-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}phenol
1-[1-(2-benzyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-4-phenylpiperazine
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-decahydro-1,6-naphthyridin-2-one
5-({[6-(dimethylamino)pyrimidin-4-yl](methyl)amino}methyl)-2-methoxyphenol
N-[(3R,4S)-4-cyclopropyl-1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]pyrrolidin-3-yl]cyclobutanecarboxamide
1-{5-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]thiophen-2-yl}ethan-1-one
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-ol
1-{2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N2-benzyl-6-(2,4-difluorophenyl)-1,3,5-triazine-2,4-diamine
(2R,3S,6R)-3-(4-methylphenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-[3-(4-cyclopropanecarbonyl-3-fluorophenyl)phenyl]ethyl}pyrrolidine
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
2-(3,4-difluorophenyl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methoxypropanamide
2-cyclobutyl-N-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-{3-[2-(3-methoxypropyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-(hydroxymethyl)-1-{[4-(2-phenylethoxy)phenyl]methyl}pyrrolidin-3-ol
N-(1-methoxypropan-2-yl)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-N-methyl-2-(3-methyl-1,2-oxazol-5-yl)acetamide
(2S,4S)-4-[4-({[(3,4-dimethylphenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
2-(dimethylamino)-8-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(3-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
4-{[5-(1-cycloheptylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
6-[2-(1-hydroxyethyl)-1-methyl-1H-1,3-benzodiazol-5-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-(azepane-1-carbonyl)-N-cyclooctyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-(2-methoxyphenyl)-2-methyl-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
2-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(piperidine-1-carbonyl)pyridine
N-{2-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
4-{1-[1-(4-chlorophenyl)cyclobutanecarbonyl]piperidin-3-yl}pyrimidine
2-(2-methylphenyl)-5-{1-[1-(1,3-thiazol-2-yl)propyl]-1H-1,2,3-triazol-4-yl}pyrimidine
N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-(trifluoromethyl)benzene-1-sulfonamide
1-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N,6-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(diethylamino)ethyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
2-{5-[1-(4-methoxy-3-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(4-methylpent-3-en-1-yl)piperazin-2-yl}ethan-1-ol
(1S,6R)-9-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
N-(pyridin-2-ylmethyl)-4-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
methyl[(3-{[1-(quinoline-8-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-2-ylmethyl)amine
2-[9-(6-methyl-2-propylpyrimidin-4-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-(1-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1H-1,2,3-triazol-4-yl)phenol
methyl 6-[(3-methylphenyl)methyl]-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate