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1-{furo[3,2-c]pyridin-4-yl}-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-(3-hydroxypropyl)-8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]propanamide
4-{3-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(3S,4S)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
5-ethyl-3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1,2-oxazole
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)but-2-ynamide
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}({[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl})amine
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
2-(3-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
7-fluoro-2-[4-(4-methoxybutyl)piperazine-1-carbonyl]-3-methyl-1H-indole
[(3-fluoro-4-methoxyphenyl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
{[1-(3-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}urea
N-methyl-3-[(1-oxo-1,2-dihydrophthalazin-2-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,3,4,7-tetramethyl-1H-indole-2-carboxamide
1-[2-(2-methoxyphenoxy)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
1-(furan-2-ylmethyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]piperidine-4-carboxamide
2-[3-(3-methoxybenzoyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
{4-[(4-methoxyphenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}methanol
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[4-(azetidin-1-yl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
2-(2,4-difluoro-3-methoxyphenyl)-1H-1,3-benzodiazole
(4aR,7aS)-1-ethyl-4-{2-methyl-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-benzyl-3-ethyl-1-(2-fluorobenzoyl)-1,4-diazepan-5-one
2,6-dimethyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)quinoline-4-carboxamide
1-{2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-[2-(4-fluorophenyl)ethyl]piperidine
N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-1H-imidazole-5-carboxamide
3-[(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)methyl]-N-methyl-1,2,4-oxadiazole-5-carboxamide
4-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-1-ethyl-1,2-dihydropyridin-2-one
8-(3-methylbut-2-enoyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
methyl 5-({3-tert-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)-1-methyl-1H-pyrrole-2-carboxylate
N-butyl-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-7-carboxamide
2-[8-(2,3-dihydro-1H-inden-2-yl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
3-(3-fluorophenyl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-(6-hydroxy-6-methylheptan-2-yl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
N-[3-(furan-2-yl)-3-phenylpropyl]pyridazine-4-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-[4-(methylsulfanyl)phenyl]ethan-1-one
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-N,N-dimethylazepan-4-amine
5-(1H-1,3-benzodiazol-1-yl)-N-(pyridin-3-yl)furan-2-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide