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1-{3-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}ethan-1-one
4-amino-2-({[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)pyrimidine-5-carbonitrile
1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-benzyl-5-[(diethylcarbamoyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-(4-phenoxybenzoyl)piperidin-1-yl]but-3-en-1-one
1-[3-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}piperidin-1-yl)phenyl]pyrrolidin-2-one
ethyl 1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazole-2-carboxylate
N-[(3R,4S)-1-acetyl-4-phenylpyrrolidin-3-yl]-4-(morpholin-4-yl)butanamide
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
3-methyl-8-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-(3-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
2-[(3aS,6aR)-3-cyclopentyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carbonitrile
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]pyrrolidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl]methanesulfonamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,5,6-trimethylpyrimidin-4-amine
2-[2-(cyclohexylamino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(2-amino-1,3-thiazol-4-yl)methyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-{2-[1-(5-fluoro-2-methoxybenzoyl)piperidin-2-yl]ethyl}morpholine
13-[2-(propylamino)pyrimidin-5-yl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
1-(6-aminopyridin-2-yl)-2-methyl-1H-1,3-benzodiazole-4-carboxylic acid
2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyridine-4-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
(1R,5R)-3-benzoyl-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-N-methyl-1,3-thiazol-2-amine
1-(carbamoylmethyl)-N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]piperidine-4-carboxamide
3-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-(4-methoxyphenyl)urea
2-{4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}pyrazine
5-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(1-cyclobutylethyl)-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
4-(1H-imidazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
1-[1-(3,3-diphenylpiperidin-1-yl)-1-oxopropan-2-yl]pyrrolidin-2-one
3-(2-methoxyethyl)-3,4-dihydroquinazolin-4-one
(1R,2S)-N-methyl-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclohexane-1-carboxamide
2-ethoxy-6-{[methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amino]methyl}phenol
N-[4-(2-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-1H-imidazol-1-yl)phenyl]acetamide
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}pyridazine-4-carboxamide
6-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl({[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}){4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
3-(2-methyl-1,3-oxazol-4-yl)-4-(3-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,4-oxazepan-6-ylmethyl)-3-phenoxybenzene-1-sulfonamide
N-[(2-chloro-6-fluorophenyl)methyl]-6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4R)-1-[3-(azocan-1-yl)propanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
2-cyclopropyl-5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-4-methylpyrimidine
3-(4-methylphenyl)-1-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propan-1-one
1-[(3-fluorophenyl)methyl]-4-[(2-methyl-1,3-oxazol-4-yl)methyl]piperazine
2-[5-(4-chlorophenyl)-1H-indazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine