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N,N-dimethyl-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azepan-4-amine
N-ethyl-4-(4-methylphenoxy)-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
5-fluoro-3-methyl-2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}-1H-indole
4-methanesulfonamido-N-(5-pentyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N'-cyclooctyl-N-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]butanediamide
5-{[(3,4-difluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{1-[(3E)-hex-3-enoyl]piperidin-4-yl}methanesulfonamide
8-(2,5-dimethylfuran-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3aR,7aS)-2-[4-(1H-imidazol-1-yl)benzoyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-[4-(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperazin-1-yl]acetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-(morpholin-4-yl)benzamide
3-(3-hydroxy-3-methylbutyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
(3R,4S)-1-[(2-methoxy-4-methylphenyl)methyl]-3,4-dimethylpiperidin-4-ol
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
4-(piperidin-4-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(4-acetylphenoxy)-N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]acetamide
1-tert-butyl-4-({[(3-fluoro-2-methylphenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
5-{imidazo[2,1-b][1,3]thiazol-6-yl}-3-(2-phenylethyl)-1H-1,2,4-triazole
1-methyl-1-[(5-methyl-1,2-oxazol-3-yl)methyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
2-{4-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]phenoxy}pyrimidine
4-{[2-(methylsulfanyl)phenyl]methyl}morpholine-2-carboxamide
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2-{4-[4-(azepane-1-carbonyl)-6-methylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
5-(phenoxymethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-3-(3-methoxyphenoxymethyl)piperidine
2-(2-{[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
2-(dimethylamino)-N-(2-ethyl-1,3-dihydroxypropan-2-yl)-2-(3-fluorophenyl)acetamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-amine
4-(7-{spiro[2.3]hexane-1-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)morpholine
2-(2-ethyl-1H-imidazol-1-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
(3S,7S)-5-(pyridine-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
[9-(butane-1-sulfonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
(1R,5R)-6-(cyclobutylmethyl)-3-[3-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
6-[(dimethyl-1,3-thiazol-5-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
2-{4-[(2-aminopyridin-3-yl)methyl]piperazin-1-yl}-N-ethylacetamide
4-benzyl-2-[(3-methoxyphenyl)methyl]morpholine
1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]acetamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-[(1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)oxy]pyridine
(3aR,7aS)-5-methyl-2-{1H-pyrrolo[2,3-b]pyridin-6-yl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropan-1-amine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyridine-2-carbonyl)piperidin-3-amine
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrrole-2-carboxamide
5-{[4-(benzyloxy)piperidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
N-propyl-N-(pyridin-3-ylmethyl)-2-(pyridin-3-yloxy)acetamide