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5-fluoro-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)pyrimidin-4-amine
1-(4-methoxyphenyl)-N,2,2-trimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]cyclopropane-1-carboxamide
methyl (2S)-1-[2-(2-chloro-6-fluorobenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carbonyl]pyrrolidine-2-carboxylate
1-[4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
5-butyl-4-[5-(hydroxymethyl)furan-2-carbonyl]-1-(3-methylphenyl)piperazin-2-one
(3aR,5R,6S,7aS)-2-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
5-cyclopentanecarbonyl-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
(3aR,6aR)-2-methyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[1-(3-methylbenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-indol-3-yl)ethyl]acetamide
9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-cyclopropyl-1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-amine
3-{4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazin-1-yl}benzonitrile
N-{2-[2-(adamantan-1-yl)acetamido]ethyl}propanamide
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]ethan-1-one
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(2,5-dimethyl-1H-pyrrol-1-yl)benzamide
[1-(1-benzofuran-5-ylmethyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
2-[4-(2,6-dimethylquinoline-3-carbonyl)morpholin-2-yl]ethan-1-amine
2-benzyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-1,3-benzoxazole
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]oxolane-2-carboxamide
N-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
6-ethyl-N-[2-(1H-imidazol-1-yl)propyl]-2-methylquinoline-4-carboxamide
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-4-methylphenol
4-{1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}benzoic acid
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
2-{1-[(5-tert-butyl-2-hydroxyphenyl)methyl]piperidin-4-yl}-N-methylacetamide
(3-benzyl-1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methanol
5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]pyrrolidin-2-one
2-(2-ethylpyrimidin-5-yl)-N,8-dimethyl-N-(propan-2-yl)quinoline-4-carboxamide
5-(methoxymethyl)-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}furan-2-carboxamide
7-(3-methylfuran-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-methyl-1,3-oxazole-4-carboxamide
4-(cyclohex-3-en-1-yl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole
ethyl 3-{[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]formamido}butanoate
2-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
1-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-cyclopentyl-4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
1-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-3-carbonitrile
[(2S)-1-{1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidine-4-carbonyl}pyrrolidin-2-yl]methanol
(4aS,7aR)-1-(3,5-dichloro-4-methylbenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2-fluoro-2-phenylacetyl)-1-(2-methylphenyl)piperazin-2-one
[2-(adamantan-1-yl)ethyl](methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[3-(furan-2-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-butyl-N-(5-carbamoyl-2-fluorophenyl)-2,5-dihydro-1H-pyrrole-1-carboxamide
{3-[(2-methylphenyl)methyl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl}methanol
3-(2,3-dihydroxypropyl)-1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-methylurea