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(3S,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-methylpiperidine-3,4-diol
4-({1-[2-(4-fluorophenoxy)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
methyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
3-{3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2,5-dimethylpyrazine
1-[2-({[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)amino)ethyl]piperidin-2-one
4-{2-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
3-(2-{cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
N,N-dimethyl-2-(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}-1,4-diazepan-1-yl)acetamide
[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl][1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
1-[(5-chlorothiophen-2-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(methyl)[2-(piperidin-1-yl)ethyl]amine
2-[2-({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)ethyl]-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
2-(2-methyl-1,3-thiazol-4-yl)-1-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethan-1-one
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}pent-4-enamide
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(pyridin-3-yl)pyridine-3-carbonitrile
N-methyl-2-(2-propyl-1H-1,3-benzodiazol-1-yl)-N-(1H-pyrazol-5-ylmethyl)propanamide
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
6-[2-(methylsulfanyl)phenyl]-9H-purine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]ethan-1-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-[(pyridin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-ol
[(3R,4R)-1-(2,5-dimethoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-methoxyquinoline-4-carboxamide
2-cyclopentyl-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
ethyl 3-[(2,4-difluorophenyl)methyl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine-3-carboxylate
2-[4-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
4-(2-methyl-1H-imidazol-1-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine-4-carboxylic acid
3-[(1,4-dioxan-2-ylmethyl)sulfamoyl]-N-ethyl-N-methylbenzamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(4-hydroxypiperidin-1-yl)ethyl]butanamide
3-(5-methylthiophen-2-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
(2S,4R)-4-amino-1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
8-(4-ethoxy-3-methylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-methyl-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
N-cyclopropyl-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](furan-2-ylmethyl)(thiophen-3-ylmethyl)amine
(3R,4S)-4-cyclopropyl-1-(quinoxaline-5-carbonyl)pyrrolidin-3-amine
3-{1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(3-hydroxy-3-methylbutyl)-N-[(1S,2R)-2-(hydroxymethyl)cyclopentyl]benzamide
2-({2-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-(6-chloro-1,3-benzothiazol-2-yl)-N-[2-(pyridin-3-yl)ethyl]piperidin-4-amine
N-(2-methoxyethyl)-7-(1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-methyl-1-(2-methylphenyl)piperazin-2-one
6-(methoxymethyl)-1-methyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S)-N-tert-butyl-2-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-{1-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol