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N-(2,3-dihydro-1-benzofuran-3-yl)-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
3-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-[6-(dimethylamino)pyridazin-3-yl]-N,N-bis(propan-2-yl)benzamide
[(4,6-dimethylpyridin-2-yl)methyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[2-(dimethylamino)-1-phenylethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-4-oxo-N-(oxolan-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)piperidine-3-carboxamide
3-({2-[1-(2-hydroxyethyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(propane-2-sulfonyl)pyrrolidin-3-amine
[(4aS,8aR)-6-[(2-cyclohexylpyrimidin-5-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
1-[3-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
4-cyclobutanecarbonyl-N-[4-(propylsulfanyl)phenyl]-1,4-diazepane-1-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-[4-(pyridin-2-yl)pyrimidin-2-yl]piperidin-4-ol
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[(3-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}piperidin-3-yl)benzoic acid
1-(3-methylbutyl)-3-(2-methylpropyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-[(5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1,2,4-oxadiazol-3-yl)methyl]piperidine
2-({1-[(2-methoxyphenyl)methyl]-6-oxopiperidin-3-yl}formamido)acetamide
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5,6-dimethylpyrimidin-4-amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl]methanol
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-propylpyrimidine-5-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
3-methoxy-5-[methyl(1-methylpyrrolidin-3-yl)carbamoyl]benzoic acid
4,5-dimethyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
6-ethoxy-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1,2-dihydroquinolin-2-one
2-[(1S,5R)-3-[(4-ethylphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
2-(propan-2-yl)-5-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]methyl}pyrimidine
5-{[4-(azocane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-2-methyl-1,3-benzothiazole
3-{5-[2-methoxy-5-(propan-2-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propanamide
3-[5-(5-amino-1H-pyrazole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopentylpropanamide
2-(1-phenyl-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H-1,2,4-triazol-3-yl)acetamide
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N'-(4-methylphenyl)propanediamide
(3R,4R)-4-amino-1-{[2-(2-phenylethoxy)phenyl]methyl}piperidin-3-ol
3-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-[2-(propylsulfanyl)phenyl]urea
4-[5-(1-benzylpyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
6-(morpholin-4-yl)-N4-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]pyrimidine-2,4-diamine
4-[3-methyl-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl]pyridine
N-[(4,6-dimethylpyridin-3-yl)methyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-N-phenylpropanamide
1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-amine
N-(2-methoxyethyl)-N-[(2-methylphenyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
6-(methoxymethyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-4-amine
6-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-[4-(oxane-4-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one