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3-{methyl[2-(1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
methyl 3-(1-benzothiophen-2-ylmethyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-(1H-indol-2-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
6-ethyl-1-methyl-N-{2-[methyl(phenyl)amino]propyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-methyl-2-({[3-(pyrrolidin-1-yl)propyl]amino}methyl)quinolin-4-ol
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1-benzothiophene-5-carboxamide
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-(1,3-thiazol-2-yl)piperazine
3-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-2-yl}-4-methyl-1,2,5-oxadiazole
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
1-{[2-(benzyloxy)phenyl]methyl}-3-methoxypyrrolidine
N-cyclopentyl-1-[1-(thiophen-3-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
(1R,5R)-N-[(2-fluorophenyl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[1-(8-chloroquinolin-2-yl)piperidin-4-yl]piperidin-3-ol
4-({[1-(2-fluorophenyl)cyclopentyl]methyl}amino)-1λ4-thian-1-one
4-({2-[(3-chloro-5-methylpyridin-2-yl)oxy]phenyl}methyl)morpholine
2-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}acetamide
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N,N-dimethylpyridine-3-carboxamide
2-{4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
1-(azepan-1-yl)-3-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}propan-2-ol
6-methoxy-1-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-indole-2-carboxamide
6-methoxy-4-(1,4-oxazepane-4-carbonyl)-1,2,3,4-tetrahydroquinolin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(1R,2R,6S,7S)-N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4R)-1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-4-methylpiperidine-3,4-diol
1-(1-{2,8-diazaspiro[4.5]decane-3-carbonyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(2S,4R)-4-amino-N-ethyl-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-2-carboxamide
2-ethyl-4-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1,3-oxazole-5-carboxamide
N-butyl-N-(furan-2-ylmethyl)-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
2-{[(3R,5S)-1-[(2,5-dimethylphenyl)methyl]-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
2-[5-(1,4-dimethyl-1H-indol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethan-1-ol
(1S,5R)-6-benzyl-3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
[(3R,5R)-1-(5-ethyl-1,2-oxazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(2-phenylethyl)-N-propylacetamide
3-(1-methylpiperidin-2-yl)-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-amino-N-ethyl-1-[3-(4-hydroxyphenyl)benzoyl]pyrrolidine-2-carboxamide
1,5-dimethyl-4-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1H-pyrazole
(4aS,7aR)-1-[(3,4-difluorophenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(diphenylmethyl)-5-(oxolane-3-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[2-(2-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-(pyrrolidin-3-yl)acetamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methyl-4-(3,4,5-trimethoxyphenyl)-5H,6H,7H-cyclopenta[d]pyrimidine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide