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1-(3-{4-[(dimethylamino)methyl]piperidine-1-carbonyl}phenyl)-4-ethyl-3-methyl-1H-pyrazol-5-ol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
methyl[3-(5-methylfuran-2-yl)butyl](4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
2-({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-3-methylbutan-1-ol
6-ethyl-N-{3-[methyl(phenyl)amino]propyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
methyl 1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-5-[(thiolan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(hydroxymethyl)-1,3-oxazolidin-2-one
3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
1-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
4-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-1-yl}quinazoline
N-(3,3-diphenylpropyl)-2-(ethylamino)pyrimidine-5-carboxamide
N-(prop-2-en-1-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N,N-dimethyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
3-[1-({3-[1-(dimethylamino)ethyl]phenyl}methyl)piperidin-4-yl]propanoic acid
6-cyclopropyl-2-[2-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
5-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyridin-2-amine
methyl 6-[(2,4-difluorophenyl)methyl]-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methyl-5-{4-[4-methyl-3-(1H-pyrrol-1-yl)benzoyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-(4-chlorophenyl)-3-[1-(dimethylsulfamoyl)piperidin-3-yl]propanamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
4-[4-ethyl-4-(hydroxymethyl)piperidine-1-carbonyl]pyridin-3-ol
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-{[5-(3-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}acetamide
1-ethyl-N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
2-(1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)benzoic acid
2,5-dioxo-6-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-methyl-6-propylpyrimidine
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
4-({[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
2-methoxy-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]acetamide
2,2,2-trifluoro-N-{2-[2-(pyridin-3-yl)acetamido]ethyl}acetamide
(3aR,6aR)-2-acetyl-5-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-fluorophenyl)-2-[5-methyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
8-(2-cyclopentylacetyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2,5-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
5-[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-ol
2-(ethylamino)-N,4-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-thiazole-5-carboxamide
5-ethyl-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
5-[1-(2,2-dimethylpropanoyl)pyrrolidin-2-yl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)thiophene-2-carboxamide
1-(cyclohexylmethyl)-N,N-dimethyl-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-ethyl-4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
3-methyl-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1-(2-methylpropyl)piperazin-2-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(pyrrolidin-3-yl)benzamide
3-(1H-indol-7-ylmethyl)-7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane
[(2S,6S)-4-(4-chloro-3-methylbenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-[(2R,3R,6R)-5-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2-(methylsulfanyl)pyridine