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2-[4-(4-propylpyrimidine-5-carbonyl)piperazin-1-yl]-1,3-benzothiazole
2-methyl-N-(oxolan-3-yl)-7-(thiophene-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-{[(cyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
(2R,3R)-3-amino-1'-(2-hydroxybenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2-fluorophenyl)methyl]-N,N-dimethylpiperidin-3-amine
3-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-1-[1-(4-methylpyridin-2-yl)propyl]urea
(3S,4R)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[2-(2-chlorophenoxy)ethyl]-N-ethyl-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-[2-hydroxy-3-(2-methoxy-4-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propyl]piperidin-4-ol
diethyl({3-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
3-[2-methyl-3-(trifluoromethyl)phenyl]-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl 2-(5-carbamoylpyridin-3-yl)benzoate
4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]-N-propylpiperidine-1-carboxamide
2-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-1,2-oxazolidine
3-[4-(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl)pyridin-2-yl]phenol
4-hydroxy-1-methyl-N-(4-phenylbutyl)piperidine-4-carboxamide
(1R,9S)-5-amino-3-[5-(2-cyanophenyl)furan-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-1,3-benzoxazole
1-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(4-fluorophenyl)ethan-1-one
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
4-[1-(4-methanesulfonylbenzoyl)piperidin-3-yl]benzoic acid
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-N-methyl-N-(thian-4-yl)butanamide
2-(4-fluorophenyl)-1-[3-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxymethyl)piperidin-1-yl]ethan-1-one
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
3-({[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
(3R,4R)-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
2-benzyl-8-[2-(methylsulfanyl)pyridine-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-chloro-5-(trifluoromethyl)benzamide
4-methyl-N-{2-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
N-[3-(furan-2-yl)propyl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
2-(dimethylamino)-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]acetamide
[3-cyclopropanecarbonyl-9-(1,3-thiazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
ethyl 4-[1-(propan-2-yl)-1H-pyrazole-4-amido]piperidine-1-carboxylate
1-(2-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
2-[2-(2-butyl-1H-imidazol-4-yl)-1H-imidazol-1-yl]-N-(2-methylphenyl)acetamide
2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)-N-[4-(3-methylphenyl)-1-phenyl-1H-pyrazol-5-yl]acetamide
2-[(2-fluorophenyl)methyl]-4-{4-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
6-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)pyridine-2-carboxylic acid
3-{3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidine-1-carbonyl}-1H-indazole
6-(2-hydroxyethyl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
ethyl 1-[3-(methylsulfanyl)propanoyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
2-[4-(oxolan-3-ylmethyl)-1,4-diazepan-1-yl]-1,3-benzothiazole
1-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]piperidine-4-carbonitrile