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3-{[(2-hydroxy-2-methylpropyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[2-(2-fluorophenyl)-1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N,2-dimethylfuran-3-carboxamide
9-ethyl-1-methyl-4-[5-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(azetidine-1-carbonyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methylbenzene-1-sulfonamide
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2,5-dimethoxyphenyl)methyl]piperidine
5-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
3-methyl-5-(1-methyl-1H-pyrazol-4-yl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
(3R,4R)-4-amino-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperidin-3-ol
5-ethyl-N-{[3-(methylsulfanyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
N-benzyl-N-methyl-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
2-(dimethylamino)-2-(4-fluorophenyl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
1-[(4-chlorophenyl)methyl]-4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazole
3-chloro-N-(3-hydroxypropyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
2-(pyridin-4-ylmethyl)-9-(4,4,4-trifluorobutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-oxoethyl)phenyl]butanamide
1-(4-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-[(1S,5R)-6-[3-(2-methoxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
6-chloro-N,1-dimethyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-indole-2-carboxamide
[(3R,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(2-methyl-1-benzothiophen-3-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
N-methyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-1,3-thiazol-2-amine
5-fluoro-2-[1-(1H-indazole-3-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2-[1-(1,3-thiazol-4-ylmethyl)pyrrolidin-2-yl]pyridine
6-fluoro-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[2-(pyridin-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-methoxy-N-({1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-4-oxo-4H-chromene-2-carboxamide
5-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-1,3-benzothiazol-2-amine
1-methyl-4-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
methyl 4-[(4-{2-[(oxolan-2-ylmethyl)carbamoyl]ethyl}piperidin-1-yl)methyl]benzoate
N-(2-methanesulfonylethyl)-2,8-dimethylquinoline-3-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
3-(oxolan-3-yl)-5-(2,3,6-trimethylphenoxymethyl)-1,2,4-oxadiazole
2-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-oxaspiro[4.5]decane-4-carboxamide
(2S,4S)-N-ethyl-1-hexanoyl-4-(4-hydroxybenzamido)pyrrolidine-2-carboxamide
(1R,9S)-5-amino-3-[4-methoxy-3-(methoxymethyl)phenyl]-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(2-methylphenyl)-4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N-ethyl-2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}pyridine-4-carboxamide
3-(3-methanesulfonamido-4-methoxyphenyl)-1-(oxan-4-yl)urea
5-[2-(difluoromethoxy)phenyl]-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
3-(4-methylphenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
1-(4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1-methylcyclopropanecarbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-chloro-3-methylphenoxy)-3-[(1-cyclopropylethyl)amino]propan-2-ol
6-(furan-3-carbonyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane