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N-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)methanesulfonamide
3-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-(oxan-4-yl)urea
3-({[1-(3-phenyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
(3S,4S)-1-(2-ethoxyethyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
2-[({5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)sulfanyl]pyrimidine
2,5-dimethoxy-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}benzene-1-sulfonamide
{1-[3-(6-methoxypyridazin-3-yl)phenyl]ethyl}dimethylamine
1-(4-cyclohexylphenyl)-3-methyl-3-[1-(1,2-oxazol-3-yl)ethyl]urea
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1H-pyrazole-3-carbonyl)piperidin-3-ol
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-(piperidin-1-yl)propanamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
3-phenoxy-N-[1-({[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
2-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[(4-methoxypyridin-2-yl)methyl]-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
6-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
5-[3-(2-aminoethyl)piperidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
2,6-dimethoxy-N-[1-(pyrimidin-4-yl)ethyl]pyridine-3-carboxamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}butanamide
9-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-7-(3-chlorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
1-(3-chloropyridin-2-yl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
1-(6-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
(3aR,5S,6S,7aS)-2-(1H-indole-6-carbonyl)-octahydro-1H-isoindole-5,6-diol
1-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
(3aS,6aS)-3a-(hydroxymethyl)-N-[3-(1,3-oxazol-5-yl)phenyl]-octahydrocyclopenta[c]pyrrole-2-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(propan-2-yl)pyrimidin-2-amine
N-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}pyrimidin-2-amine
2-(2-{[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]methyl}-4-(pyridin-2-yl)phenoxy)acetic acid
4-(2-{[1-(propan-2-yl)piperidin-3-yl]formamido}ethyl)benzoic acid
5-[4-(trifluoromethyl)pyridin-2-yl]-1,2,3,4-tetrahydroisoquinoline
ethyl 2-[1-(cyclohex-3-en-1-ylmethyl)-4-(4-fluorobenzenesulfonyl)piperidin-4-yl]acetate
3-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
2-({1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
1-[cyclohexyl(methyl)amino]-3-[3-({[(2,6-difluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
2-(1-methyl-1H-indol-3-yl)-1-[4-(pyridin-4-yl)piperidin-1-yl]ethan-1-one
N-cyclopropyl-4-methoxy-2-[(1-methylpiperidin-4-yl)oxy]benzamide
3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-8-(quinoxalin-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-fluorophenyl)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
7-{2-[3-(trifluoromethyl)phenyl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one