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N-[(3R,4S)-4-(propan-2-yl)-1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]furan-2-carboxamide
N,2,5-trimethyl-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
[(2-butyl-1H-imidazol-4-yl)methyl](ethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
5-[3-(3-methylphenoxy)azetidin-1-yl]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(3-methylphenyl)ethyl]piperidine-3-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2,3,6-trimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
1-[3-(3,4-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine
1-(cyclopentylcarbamoyl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-{1-[4-(morpholin-4-yl)butanoyl]piperidin-3-yl}benzoic acid
3-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
methyl 4-{[(1S,4S)-5-(5-chloro-2-methoxyphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}benzoate
2-amino-7-(5-phenoxyfuran-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-cyclohexyl-3-[2-(methylsulfanyl)benzoyl]piperidine
4-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2-(trifluoromethyl)morpholine
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-methylfuran-3-carboxamide
4-(1-hydroxy-3-methylbutyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
3-fluoro-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}pyridine
(1s,4s)-4-{4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
3-methoxy-2-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenol
N-[3-(cyclohexyloxy)-2-hydroxypropyl]-2-(4-propanoylphenoxy)acetamide
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3-phenylcycloprop-2-ene-1-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
4-(2-chloro-4-fluorophenyl)-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
(1S,5R)-6-[3-(methylsulfanyl)propyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-({4-[1-(oxan-4-yl)piperidine-4-carbonyl]piperazin-1-yl}methyl)phenol
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
8-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carboxamide
[(2S)-1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}pyrrolidin-2-yl]methanol
6-methoxy-3-methyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1-benzofuran-2-carboxamide
(1R,5R)-3-(2-methyl-4-phenylpyrimidine-5-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
4-({2-[1-(5-chlorothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(2-methylpyrrolidin-1-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
4-(1-butyl-1H-imidazol-2-yl)-N-[(3-fluorophenyl)methyl]piperidine-1-carboxamide
3-(2,3-dihydroxypropyl)-5-(3,4-dimethoxyphenyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
dimethyl({4-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)amine
N-(1-ethyl-5-oxopyrrolidin-3-yl)-3,6-dimethyl-1-benzofuran-2-carboxamide
N-methyl-7-oxo-N-[(1-phenylpyrrolidin-3-yl)methyl]-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]urea
{4-[(3-methoxyphenyl)methyl]-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl}methanol
4-methyl-N-[(2-methylpyridin-4-yl)methyl]-3-(2-oxoimidazolidin-1-yl)benzamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(morpholin-4-yl)ethyl]amine
1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
6-methyl-N-{2-[1-(pyridin-4-ylmethyl)piperidin-3-yl]ethyl}pyridine-2-carboxamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(4-methylnaphthalene-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-propylpyrrolidin-3-yl]pyridine-2-carboxamide