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2-{4-[1-(4-chlorophenyl)piperidin-4-yl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
3-[(3R,4S)-1-(2-methyl-1H-pyrrole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-{2-[methyl(2-phenylethyl)amino]ethyl}-8-propanoyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl(oxolan-3-ylmethyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
7-(4-methyl-1H-imidazole-2-carbonyl)-N-(oxolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-9H-purin-2-amine
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-cyclopropyl-1H-pyrazole
2-[5-benzyl-4-(2-ethoxyacetyl)-2-oxopiperazin-1-yl]benzonitrile
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
N-(2-hydroxyethyl)-N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-yl}piperazine
4-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}thiomorpholine
1-(cyclobutylmethyl)-3-hydroxy-3-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)piperidin-2-one
N-(propan-2-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
4-(4,4-difluoropiperidine-1-carbonyl)-N-methylpyridin-2-amine
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-1,4-oxazepane
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylpyridine-3-carboxamide
2-(1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
1-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-3-(4-methylphenoxymethyl)piperidine
N-cyclopropyl-2-(2,4-difluorophenoxy)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-(3-fluorophenyl)-N-{[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
2-{[(4-fluorophenyl)methyl]({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})amino}butan-1-ol
2-methoxy-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-5-sulfamoylbenzamide
3-(3-fluorophenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-2-one
(1-{1-[1-(3-methoxyphenyl)piperidin-4-yl]piperidin-3-yl}piperidin-4-yl)methanol
8-(4-methyl-1H-imidazole-5-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-(4-{2-[(4aR,8aR)-6-(3-methylbutyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methoxypiperidine
N-phenyl-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]propanamide
6-methyl-2-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyridine-3-carboxamide
N-methyl-2-(1H-pyrazol-1-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
2-[(3-methylpiperidin-1-yl)methyl]-4-(pyridin-3-yl)phenol
[4-({3-[(furan-2-ylmethyl)sulfanyl]propyl}amino)quinazolin-2-yl]methanol
2,3,5,6-tetramethyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}benzamide
3-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-2,6-dimethyl-1,4-dihydropyridin-4-one
N-(2-methoxyethyl)-4-methyl-3-{[(oxan-4-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-cyclopropanecarbonyl-1'-(2-methoxypyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
3-[(3R,4S)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-ethyl-8-[(3-methyl-1H-indol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(1-ethylpiperidin-3-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
2-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine-3-carbonyl}pyridine
methyl 4-{[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]amino}-3-chlorobenzoate
3-[4-(hydroxymethyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
3-(3-chloro-1,2-oxazol-5-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-{2-[2-(propylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethan-1-ol
N-(2-methoxyethyl)-5,6-dimethyl-N-(thiophen-3-ylmethyl)pyridine-3-carboxamide