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(2S,4S)-4-{[(4-chlorophenyl)methyl]amino}-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
methyl 4-({1-ethyl-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl}methyl)benzoate
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
N-[(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)methyl]methanesulfonamide
1-(furan-2-ylmethyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]piperidine-4-carboxamide
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
7-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
2-{4-[2-(1H-imidazol-2-yl)benzoyl]piperazin-1-yl}pyridine-3-carbonitrile
1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-[2-(5-methylthiophen-2-yl)ethyl]urea
3-(oxolan-3-yl)-5-(3-phenylpropyl)-1,2,4-oxadiazole
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-fluorophenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
8-(2-methoxyacetyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(piperidin-1-yl)acetamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
2-(methylamino)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyridine-4-carboxamide
N-(pyridin-3-ylmethyl)-1-{1-[2-(pyrrolidin-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
methyl 3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
2,6-dimethoxy-4-(4-phenyl-1H-imidazol-5-yl)phenol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
3-methyl-1-{4-[5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]phenyl}-1H-pyrazol-5-amine
4-(2-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-2-yl}ethyl)morpholine
6-(4-methanesulfonylphenyl)hexan-1-ol
2-tert-butyl-5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-1,3,4-oxadiazole
2,3-dimethyl-6-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N-benzyl-2-butyl-2,5-dihydro-1H-pyrrole-1-sulfonamide
2-(morpholin-4-yl)-N-[2-(phenylsulfanyl)ethyl]-2-(pyridin-3-yl)acetamide
3-(3-methoxyphenyl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-5-carboxamide
N-benzyl-1-[1-(cyclopentylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[4-oxo-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]benzonitrile
3-fluoro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyridine-4-carboxamide
1-(4-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
4-{2-[4-(1,3-thiazole-4-carbonyl)morpholin-3-yl]acetyl}-1λ6-thiomorpholine-1,1-dione
N-[2-(4-methoxyphenyl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxamide
1'-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2-hydroxypyridin-3-yl)acetamide
4-[(2S,3R)-2-amino-3-hydroxybutanoyl]-1-(2-methylphenyl)piperazin-2-one
3-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
N-methyl-3-({[1-(pyridin-3-ylmethyl)piperidin-4-yl]carbamoyl}amino)benzamide
2-(5-acetylthiophen-3-yl)-1-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
methyl 5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}methanesulfonamide
1-cyclopentyl-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
(3S,4R)-1-[4-(azepan-1-yl)-4-oxobutanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
4-[1-cyclohexyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carbonyl]-1-phenylpiperazin-2-one
ethyl 3-benzyl-1-[(2,3-dimethylphenyl)carbamoyl]piperidine-3-carboxylate
N'-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-N-(propan-2-yl)ethanediamide