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5-(methoxymethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylfuran-2-carboxamide
N-(2-methoxyethyl)-5-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-ethyl-6-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-methylpyrimidin-4-amine
2-(4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
1,3-dimethyl-5-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-{1,4-diazabicyclo[3.2.2]nonan-4-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
2-{[(1-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)oxy]methyl}pyridine
1-(2-methoxyphenyl)-4-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]piperazine
[2-(1-{1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-2-yl)ethyl]dimethylamine
8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(4-methoxypiperidin-1-yl)pyridine
5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-pyrazole
2-(dimethylamino)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-6-(2-methylphenyl)pyridine-3-carboxamide
2-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
5-(3-acetylphenoxymethyl)-N-(1-methoxybutan-2-yl)-1,2-oxazole-3-carboxamide
1-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-(5-methyl-2,1,3-benzothiadiazol-4-yl)urea
N-(3,4-difluorophenyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-amine
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyridin-2-yl)propan-1-one
1-{3-oxo-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propyl}piperidin-2-one
3-(3-fluoro-4-phenylbenzoyl)-1-methylpiperidine
N,1-dimethyl-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-3-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(3-methylpyridin-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
5-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-(4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazin-1-yl)-1,3-benzothiazole
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxybenzamide
(1R,2S,6R,7S)-4-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
N4-(2-methoxyethyl)-7-(1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-({5-fluoro-2-[3-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-{[4-(1-propyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
2-{3-cyclopropyl-5-[2-(2-methoxyphenyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
[(4-fluorophenyl)methyl](methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1-[4-(piperidin-3-yl)benzoyl]piperidine
2-{5-[2-(phenylamino)pyrimidine-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
4-{3-[1-(2-fluoroethyl)-1H-pyrazol-3-yl]phenyl}-N,N,6-trimethylpyrimidin-2-amine
1-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidine-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(propan-2-yl)pyrimidine-4-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-4-carboxamide
1-methyl-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-(1,2,3,4-tetrahydronaphthalen-1-yl)urea
6-(1H-indol-3-yl)-2-[3-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
5-ethyl-N,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]pyrimidin-4-amine
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
4-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]-2-methoxyphenol
4-{[4-(furan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-2-methyl-1,4-diazepan-5-one
3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-4-methylpyridine
8-(2,2-dimethylpropyl)-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione