Tips: Press Ctrl key to select multiple functional groups
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
ethyl 1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpiperidine-4-carboxamide
N-(2-{[(2-fluorophenyl)methyl]sulfanyl}phenyl)-6-hydroxy-1,4-oxazepane-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-butyl-N,5-dimethyl-1H-pyrazole-4-carboxamide
2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-[(4,4-difluoropiperidin-1-yl)methyl]-8-fluoroquinolin-4-ol
1-{2-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]phenyl}ethan-1-one
2-(cyclohex-1-en-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
1-ethyl-3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-3-(2-methylphenyl)pyrrolidin-3-ol
methyl 2-{1-[(3-methyl-1,2,4-thiadiazol-5-yl)carbamoyl]-3-oxopiperazin-2-yl}acetate
(3R,4R)-1-[(3,4-dimethylphenyl)methyl]-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
5-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
3-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-[2-(trifluoromethyl)phenyl]urea
4-(2-fluoro-6-methoxyphenyl)-2-methyl-1H-imidazole
1-(azepan-1-yl)-3-(2-methoxy-4-{[(2-methoxyethyl)amino]methyl}phenoxy)propan-2-ol
3-(3-fluoro-4-methoxybenzoyl)-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine
(1-{[1-(cyclopropanesulfonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-benzyl-1-(4-chlorophenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
(4aR,7aS)-1-acetyl-4-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-N-ethyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]pyrrolidine-2-carboxamide
(2R,3S,6R)-5-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,3-dihydro-1,2-benzothiazol-3-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-pyrazol-1-yl)butan-1-one
3-(2-chlorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-2-(2-oxoazepan-1-yl)acetamide
N-(2-{[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
2-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3-thiazole-4-carboxamide
N-(1-cyclopropylethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
(2S)-2-acetamido-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]propanamide
1-(5-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl)butan-2-ol
3-{5-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
3-methoxy-N-(1-{7-[2-(4-methoxyphenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)propanamide
4-benzyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidine
4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2-(trifluoromethyl)morpholine
4-ethyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-1,2,3-thiadiazole-5-carboxamide
5-acetyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}thiophene-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-3-amine
1-(3-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
(1R,9S)-5-amino-3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})amine
N-[2-(2,4-difluorophenyl)-1-{1-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-(azepan-1-yl)-3-[2-methoxy-4-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-(2-aminoethyl)-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-{4-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
4-chloro-1-ethyl-N-[(3R)-piperidin-3-yl]-1H-pyrazole-3-carboxamide