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N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
6-(2-aminoethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-2-methylpyrimidin-4-amine
ethyl 1-[(3-fluorophenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
N-ethyl-N-[1-(4-methoxyphenyl)propan-2-yl]-2,4-dimethylpyrimidine-5-carboxamide
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[(thiophen-2-ylmethyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-(2,4-difluorophenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
1-(furan-2-carbonyl)-4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-3-enamide
N-[(2-chlorophenyl)methyl]-3-(N-methylmethanesulfonamido)-N-(prop-2-en-1-yl)propanamide
2-(3-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
1-methyl-3-{[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(2-fluorophenyl)-4-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}piperazine
4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyridine
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(pyrrolidine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
({4-[1-(2,4-difluorobenzoyl)piperidin-2-yl]phenyl}methyl)dimethylamine
N-({5-[(4-methyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-(5-methyl-2-pentanamidophenyl)pyrazolo[1,5-a]pyridine-2-carboxamide
(1,4-dioxan-2-ylmethyl)(methyl)[(5-propylfuran-2-yl)methyl]amine
2-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,4-diazepan-6-yl}acetic acid
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
2-[(3S)-3-hydroxy-3-phenylpropyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
2-(furan-2-yl)-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-oxoacetamide
2-[3-(dimethylamino)propyl]-9-(3-hydroxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-phenyl-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecane
11-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
7-(oxan-4-yl)-2-[(5-propylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2-chlorophenyl)-1-methyl-3-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)pyrrolidine-2,5-dione
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}acetamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-(3,4-difluorobenzoyl)piperidine
N-cyclopropyl-5-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-methyl-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
2-methyl-4-(4-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}phenyl)but-3-yn-2-ol
N-(2-methoxy-6-methylphenyl)-2-(pyrrolidin-1-ylmethyl)piperidine-1-carboxamide
3-({[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
N-[1-(2-chlorophenyl)ethyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
(3aR,6aR)-2-(tert-butylcarbamoyl)-5-(propan-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-(thiophen-3-ylmethyl)piperidin-3-ol
3-(3-hydroxyquinoxalin-2-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N-(3-methoxyphenyl)-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]propanamide
2-{4-[(6-ethoxypyridin-3-yl)methyl]piperazin-1-yl}-3-methylpyrazine
N-ethyl-N-(2-methylphenyl)-3-{[2-(morpholin-4-yl)ethyl]amino}propanamide
5-[4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxymethyl]furan-2-carboxylic acid
1-[(2-fluorophenyl)methyl]-N-methyl-N-[4-(morpholin-4-yl)butyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-1-[3-(2-methylpiperidin-1-yl)propyl]-1H-1,3-benzodiazole
(3S,4S)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methoxyethyl)piperazine
1-(2-methoxy-6-{[(3-phenylpropyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-4-(methoxymethyl)-5-methyl-1,2-oxazole