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1-(1-methylcyclopropanecarbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[2-methyl-4-(propylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
(3S,4R)-4-(2-methylphenyl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
4-(2,6-dimethylquinoline-4-amido)oxane-4-carboxylic acid
2-fluoro-N-{3-oxo-3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propyl}benzamide
3-(2-methoxyethyl)-1-[(5-propylfuran-2-yl)methyl]piperidine-3-carboxylic acid
N-methyl-2-(3-{[(2-methylpropyl)(pyridin-2-ylmethyl)carbamoyl]amino}phenyl)acetamide
N-({5-[(3-methylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
1-{2-[benzyl(methyl)amino]-6-phenylpyridine-3-carbonyl}-N,N-diethylpiperidine-3-carboxamide
4-ethyl-1-methyl-3-{1-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[(3-methylthiophen-2-yl)sulfonyl]pyrrolidin-3-yl]acetamide
(1R,5R)-3-(2-methyl-1-benzofuran-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
(2S,4R)-1-benzyl-4-{[(2,6-difluorophenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
3-(propan-2-yl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
7-[(3,4-difluorophenyl)methyl]-2-(pent-4-enoyl)-2,7-diazaspiro[4.5]decan-6-one
3-{[(1-benzyl-1H-imidazol-2-yl)methyl]amino}pyrazine-2-carbonitrile
5-[(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)amino]-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}pyrazine-2-carboxamide
[(6-ethoxypyridin-3-yl)methyl](methyl)(quinoxalin-2-ylmethyl)amine
2-(dimethylamino)-N-(2-ethoxyethyl)-2-(2-fluorophenyl)acetamide
N,N,2-trimethyl-7-(2-oxo-1,2-dihydroquinoline-4-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N4-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-2,4-diamine
4-[4-(3-aminopentan-3-yl)-1H-1,2,3-triazol-1-yl]-N-[(1S)-1-phenylethyl]piperidine-1-carboxamide
3-chloro-4-fluoro-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1-benzothiophene-2-carboxamide
3-phenyl-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperazine
2-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2-dihydrophthalazin-1-one
1-methyl-6-propyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-methylthiophene-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea
2-[(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)oxy]pyrimidine
N-[(6-chloropyridin-3-yl)methyl]-1-cyclopentanecarbonyl-N-methylpiperidine-4-carboxamide
(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
methyl 2-[3-oxo-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-8-yl]acetate
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-1,4-diazepan-2-one
N-(2,4-dichloro-3-methylphenyl)-3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
5-(1,4-dioxan-2-yl)-1-[(3-methylphenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
1-methyl-4-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
3-(2-oxo-2-{4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(thiophen-2-ylmethyl)piperazine
(2S,4R)-N,N-diethyl-4-[4-(3-methoxyphenyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
(4aS,7aR)-1-(5-acetylthiophene-2-carbonyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-hydroxyphenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]propanamide
methyl(1,2-oxazol-5-ylmethyl){[5-(propane-1-sulfonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine