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3-butyl-1-methyl-4-[2-(thiophen-3-yl)acetyl]piperazin-2-one
1-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-(1H-imidazol-4-yl)ethan-1-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3,5-dimethyl-N-(oxolan-2-ylmethyl)-1,2-oxazole-4-sulfonamide
{5-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-2-fluorophenyl}methanol
ethyl 5-{[2-(5-carbamoylthiophen-2-yl)pyrrolidin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
1-({[2-(2-methoxyphenyl)ethyl]carbamoyl}methyl)piperidine-3-carboxamide
ethyl 4-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)piperazine-1-carboxylate
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)urea
N-(3-cyano-4-ethoxyphenyl)-3-(methanesulfonylmethyl)piperidine-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}pyrrolidine-2-carboxamide
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]prop-2-en-1-one
(1-benzothiophen-5-ylmethyl)(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]pyrrolidin-2-yl}-N-(1-methyl-1H-pyrazol-4-yl)thiophene-2-carboxamide
N-cyclopentyl-4-(4-{[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]amino}piperidin-1-yl)benzamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-amine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{[(3R)-3-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-(pyridin-2-yl)acetamide
4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
1-(4-chlorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclobutane-1-carboxamide
3-[3-cyclopropyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]propanamide
9-[(5-ethylpyridin-2-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-methoxy-N-({5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
[2-({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}oxy)ethyl]dimethylamine
2-(5-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1-methyl-1H-imidazole
(3-{2-[1-(3-ethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-(diphenylmethyl)-4-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]piperazine
N-cyclohexyl-2-ethyl-N-[2-(ethylsulfanyl)ethyl]-4-methyl-1,3-oxazole-5-carboxamide
N-(2-methoxyphenyl)-2-(2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-4-phenylphenoxy)acetamide
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxypropan-1-one
methyl 1-{3-[4-({[(4-fluorophenyl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
4-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-(3-chloro-4-fluorophenyl)-2-[4-(2-methoxyethoxy)piperidin-1-yl]acetic acid
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-(1-propylpiperidin-4-yl)piperidin-4-amine
9-(2-ethylpyrimidine-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-cyclohexyl-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}piperidine-4-carboxamide
N-methyl-5-({[4-(piperidin-3-yl)phenyl]formamido}methyl)furan-2-carboxamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-phenylethyl)acetamide
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
N-[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)methyl]thiophene-2-sulfonamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(2-hydroxy-5-methoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1,3-dimethyl-2,6-dioxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]sulfamoyl}-N-(2-methylpropyl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-N-(propan-2-yl)pyrimidin-4-amine
4-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-1-(3-methoxyphenyl)piperazin-2-one
1-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-ethylbutan-1-one
N-[(3R,4R)-1-[(2-chloro-4-fluorophenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
5-chloro-2-methoxy-4-({3-[(4-methoxyphenyl)amino]piperidin-1-yl}methyl)phenol
(1R,3S)-3-[1-(2,3-dihydro-1H-inden-2-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]cyclopentan-1-amine
N-(2-methyl-1-{7-[2-(methylsulfanyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)propanamide