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6-(1H-1,3-benzodiazole-5-carbonyl)-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(3-phenylpyrrolidin-1-yl)ethan-1-one
3-[5-(8-hydroxyquinoline-7-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
5-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)carbamoyl]thiophene-2-carboxylic acid
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)acetamide
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(1-methylcyclopropyl)propan-1-one
(2R,6S)-2,6-dimethyl-4-{[3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}morpholine
N-[1-(pyridin-2-yl)propan-2-yl]-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[3-(3-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1-phenylpyrrolidine
3-[2-(3,4-difluorophenyl)ethyl]-1-(3-methyl-1H-pyrazole-4-carbonyl)piperidine
4-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine
3-[2-({1-azabicyclo[2.2.2]octan-3-yl}amino)phenyl]-1,3-oxazolidin-2-one
(2R)-3-(benzyloxy)-2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)propan-1-ol
2-amino-4-(2-methoxypyrimidin-5-yl)-6-[2-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
2-(dimethylamino)-2-(3-fluorophenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
2-(phenylamino)-N-[2-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
4-{5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridine
(4S,6R)-6-methyl-N-[3-(2-phenylacetamido)phenyl]-2-sulfanylidene-1,3-diazinane-4-carboxamide
4-{1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[5-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[(1,2-oxazol-5-ylmethyl)sulfamoyl]benzamide
N-cyclopentyl-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-methoxy-1-{2-oxo-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]ethyl}-1,2-dihydropyridin-2-one
(adamantan-1-ylmethyl)({[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
4-chloro-5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
8-[2-(3-chloro-4-hydroxyphenyl)acetyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2-(4-ethoxyphenyl)-N-methylacetamide
(2R)-N-(isoquinolin-5-ylmethyl)-N-methyloxolane-2-carboxamide
2-[(cyclopropylmethyl)sulfanyl]-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
1-(4,4-difluoropiperidin-1-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
(2E)-4-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]pent-2-enamide
8-(1H-imidazol-2-ylmethyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}propan-1-ol
2-(butylsulfanyl)-N4-(oxolan-3-yl)pyrimidine-4,6-diamine
6-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
(3S,4R)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-ethyl-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
1-{1-[6-(methoxymethyl)pyridine-2-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(morpholin-4-yl)acetamide
N-[2-(diethylamino)ethyl]-5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3R,9aR)-8-(3-chlorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(4-methyl-2-oxo-2H-chromen-7-yl)-3-propylurea
1-(2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)pyrrolidin-2-one