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4-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-cyclohexyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
6-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yl)pyrimidin-4-amine
N4,N4,N6-trimethyl-N6-[(3-methylthiophen-2-yl)methyl]pyrimidine-4,6-diamine
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-methoxyphenol
N-cyclohexyl-8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
8-(2,5-dimethylfuran-3-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
1-cyclopentanecarbonyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]piperidine-4-carboxamide
N-butyl-3-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}benzamide
(3E)-1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pent-3-en-1-one
2-[methyl(pyridin-3-ylmethyl)amino]-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]propanamide
6,6-dimethyl-N-(oxan-4-yl)-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-fluoro-5-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]benzonitrile
2,3,6-trimethyl-4-(2-phenylazetidine-1-carbonyl)quinoline
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]ethan-1-one
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(2-fluorophenoxy)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
4-(1-benzyl-1H-imidazol-2-yl)-1-(1,3-thiazole-4-carbonyl)piperidine
2-(dimethyl-1,2-oxazol-4-yl)-N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
3-(1H-1,3-benzodiazol-2-yl)-N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)propanamide
3-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-4-methoxyphenol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[3-(pyridin-2-yl)propanoyl]piperidin-3-yl]propanoic acid
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-2-(1H-indol-1-yl)ethan-1-one
4-[(2-hydroxypropyl)amino]-N-[2-(1H-imidazol-4-yl)ethyl]pyridine-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}acetamide
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(1,2,4-oxadiazol-3-yl)piperidine
N-(1-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
1-[4-(2-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}ethyl)piperazin-1-yl]propan-1-one
4-acetyl-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
N-methyl-6-[(3-methylphenyl)methyl]-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-hydroxyethan-1-one
2-(2-methoxyethyl)-8-(pyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(5-butylthiophen-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane
4-(1-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}piperidin-3-yl)benzoic acid
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(3,5-difluorophenyl)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
4-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
6-fluoro-2-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methylpropanamide
7-(2,3-dimethoxyphenyl)-4-[(4-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[5-(3-methyl-2-phenylbutanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-(2-fluoroethyl)-4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2,3-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]quinoxaline-6-carboxamide
1-(4-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one