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N-benzyl-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-sulfonamide
ethyl 4-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}piperidine-1-carboxylate
N-cyclopropyl-6-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-4-[3-(oxolan-3-yl)-1-phenyl-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-amine
6-chloro-1-methyl-N-[3-(methylsulfanyl)propyl]-1H-indole-2-carboxamide
6-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)pyridine-3-carbonitrile
3-(2-fluoro-4-methoxyphenyl)-4-(1H-imidazol-2-yl)-1-phenyl-1H-pyrazole
5-(butoxymethyl)-1-(3-methylphenyl)-1H-1,2,4-triazole
6-{[1-(4-fluorophenyl)piperidin-4-yl]amino}-2-methylheptan-2-ol
4-[1-(2-ethylbenzoyl)pyrrolidin-3-yl]benzoic acid
2-ethyl-9-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N4-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
5-methyl-N-({6-methyl-2-[methyl(1H-pyrazol-5-ylmethyl)amino]quinolin-3-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
1-(4-{2-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
2-amino-4-(5-methylthiophen-2-yl)-6-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
ethyl 1-[2-(1H-imidazol-2-yl)benzoyl]-3-(2-phenylethyl)piperidine-3-carboxylate
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
N-[3-(methylsulfanyl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)-N,N-diethylpyrrolidin-3-amine
1-(2-{[(adamantan-1-yl)amino]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(azepan-1-yl)-4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}butane-1,4-dione
3-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}benzoic acid
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-methyl-N-(2-oxoazepan-3-yl)-1-benzofuran-7-carboxamide
(1s,4s)-4-{4-[3-(2-hydroxyethoxy)phenyl]-1H-1,2,3-triazol-1-yl}cyclohexane-1-carboxylic acid
3-{3-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]phenyl}-2H-chromen-2-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-oxo-2-(thiophen-2-yl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenylpropanamide
8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(furan-2-carbonyl)-1-methyl-4-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
4-(pyridin-4-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
5-(3-methyl-1,2-oxazol-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-methoxy-3-methyl-2-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-indole
2-[3-cyclopropyl-5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-[(2R)-1,1,1-trifluoro-3-methylbutan-2-yl]quinoxaline-5-carboxamide
1-{[({4-[3-(azocan-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}cyclohexan-1-ol
9-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-[2-(benzenesulfonyl)ethyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1R,3R)-3-aminocyclopentyl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanamide
4-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
5-(2-acetylphenyl)-N-tert-butylfuran-2-carboxamide
1-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]urea
3-(4-methoxyphenyl)-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-pyrazole-5-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(dimethyl-1,2-oxazol-4-yl)-3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzamide
1-ethyl-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-pyrazole-5-carboxamide
1-(3-methoxyphenyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]piperazine
methyl 2-{[2-(furan-2-yl)azepan-1-yl]methyl}-1,3-oxazole-4-carboxylate
1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol