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3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidine
N-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-ethyl-4-({methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
2-(2,5-dimethylphenyl)-1-[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]ethan-1-one
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
methyl 4-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-oxobutanoate
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2,2-diphenylacetamide
1'-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]spiro[indene-1,4'-piperidine]
3-(4-fluorophenoxy)-1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}azetidine
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
({4-cyclopropyl-5-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
({5-ethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
6-ethoxy-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
8-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
6-butyl-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
6-(3-fluoro-4-methoxyphenyl)-N,N-dimethylpyrazin-2-amine
1-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
5-(2-phenoxyacetyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(3R)-1-({1-[1-(5-methyl-1,3-benzoxazol-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-3-amine
{1-[(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
1-(3,4-dimethoxybenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}benzoic acid
3-[(4-fluorophenyl)methyl]-5-[1-(2-hydroxyethyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
[3-propyl-1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]methanol
4-[(5-ethylpyridin-2-yl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-benzyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-5-(thiophen-2-yl)benzoyl]piperazine
N-methyl-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyrazin-2-ylmethyl)pyridin-2-amine
7-(cyclohexylmethyl)-2-(ethanesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-methoxyphenyl)ethyl]-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-cyclohexyl-N-[2-(2-fluorophenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-methoxy-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(morpholin-4-yl)propan-2-yl]amine
1-{1-[(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-(2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydroisoquinolin-1-one
1-(3-chloro-4-fluorophenyl)-4-(oxolane-3-carbonyl)piperazine
8-chloro-2-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)quinolin-4-ol
7-methyl-4-(3-methylpiperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-methoxy-3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
2-(2-{[ethyl(propan-2-yl)amino]methyl}phenyl)-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
N-cyclooctyl-4-[3-(diethylamino)pyrrolidin-1-yl]-4-oxobutanamide
3-(3-hydroxy-3-methylbutyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]benzamide
(3R)-1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazine
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(pyridin-2-yl)acetamide
4-[(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
2-amino-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,6-dimethylpyrimidine-4-carboxamide
N-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
7-(cyclohexylmethyl)-2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one