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4-(4-chlorophenyl)-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}butanamide
2-(dimethylamino)-N-[(2-hydroxyadamantan-2-yl)methyl]-2-(4-methylphenyl)acetamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(3,4,5-trimethoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-hydroxy-3-({4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}methyl)-1-(2-phenylethyl)piperidin-2-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]propan-1-ol
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-methyl-2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}methyl)-1H-1,3-benzodiazole
(2R,3R,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]benzamide
2-acetamido-N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)acetamide
N-(2-methoxyethyl)-5-phenyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(pyridin-2-yl)propanoyl]-1,4-diazepan-2-one
2-(3-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
3,5-dimethyl-6-(3-methyl-1,2,4-oxadiazol-5-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-{5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
N-cyclobutyl-3-[(cyclopropylmethyl)(2-methoxyethyl)sulfamoyl]benzamide
1-(4-{[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}thiophen-2-yl)ethan-1-one
2-[3-(1,3-dimethyl-1H-pyrazol-4-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-methyl-2-[methyl(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amino]acetamide
4-methoxy-N-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-(2-methylpropyl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
6-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
N-(1,4-oxazepan-6-ylmethyl)-2-(trifluoromethyl)benzene-1-sulfonamide
2-(6-methoxynaphthalen-2-yl)-4-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]morpholine
3-{[1-(oxan-4-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
(2S,4S)-4-amino-N,N-diethyl-1-(4-methyl-1H-imidazole-2-carbonyl)pyrrolidine-2-carboxamide
3-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-1,3-diazinane-2,4-dione
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(piperidin-4-yl)pyridin-2-amine
4-amino-3-hydroxy-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}butan-1-one
N-methyl-N-[2-(morpholin-4-yl)propyl]-1-(pyridine-2-carbonyl)piperidin-4-amine
(4S)-3-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-4-phenyl-1,3-oxazolidin-2-one
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(piperidine-1-carbonyl)piperidine
3-(5-{[methyl(oxan-2-ylmethyl)amino]methyl}thiophen-2-yl)prop-2-yn-1-ol
4-chloro-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1H-pyrrolo[2,3-b]pyridine
methyl 2-(2-{[(1-ethyl-3-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
1-(2-{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-(4-chloro-2-methylphenyl)-3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-methylurea
N-(4-ethoxyphenyl)-2-(pyridin-2-yl)piperidine-1-carboxamide
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
1-cyclopentyl-5-(5-methylfuran-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methoxypropan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-methyl-1H-indole-2-carboxamide
(4aS,8aR)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-[(3-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
6-(5-chloro-2-ethoxyphenyl)pyrazine-2-carboxylic acid