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(3R,4R)-1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-(morpholin-4-yl)-1-[4-(oxan-4-yl)piperazin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-methyl-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-(azepan-1-yl)-3-{3-[(4-methylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
3-({ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenol
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(prop-2-en-1-yl)acetamide
5-(4-methoxy-2,6-dimethylphenyl)pyrazin-2-amine
2-ethyl-9-(1-methyl-1H-pyrazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-(3-{[(adamantan-2-yl)amino]methyl}-5-(pyrrolidine-1-carbonyl)phenyl)pyridine-2-carboxamide
2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylacetamide
4-(2-methoxy-2-phenylacetyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[1-(8-chloroquinolin-2-yl)piperidin-4-yl]piperidin-4-ol
2-(4-{[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidine
N-(oxolan-3-yl)-3-[(2-phenylethyl)sulfamoyl]benzamide
6-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-5,6-dihydro-1,6-naphthyridin-5-one
3-{[(3R,4S)-3-(2-carboxyethyl)-4-(dimethylamino)piperidin-1-yl]methyl}benzoic acid
2-cyclobutyl-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
N-[3-(3-methylphenyl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-3-carboxamide
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-[2-(morpholin-4-yl)ethyl]urea
7-(2,2-dimethylpropyl)-2-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
N-(propan-2-yl)-1-{1-[2-(pyridin-4-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
2-[benzyl(methyl)amino]-1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]ethan-1-one
2-(pyrrolidin-3-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]benzamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
4-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}quinoline
(2S,4S)-4-amino-N-ethyl-1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)pyrrolidine-2-carboxamide
9-(2-ethylpyridine-4-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(propan-2-yl)-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
1-(2-{[({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(pyrrolidin-2-yl)-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]thiophene-2-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methylacetamide
N4-{[4-(morpholin-4-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(1H-indol-3-ylmethyl)-N5-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-(4-{[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}piperidin-1-yl)ethan-1-one
2-methoxy-1-[1'-(3-propyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-{[4-(2,2-dimethoxyethyl)piperazin-1-yl]methyl}-1-methyl-1H-indole
4-(2-methyloxane-2-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
3-(1H-imidazol-2-yl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
ethyl 1-[(2,3-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
2-{[4-(2-chlorophenyl)-5-(1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-(1,3-benzothiazol-2-ylmethyl)-5-(methoxymethyl)-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
dimethyl({4-[2-(pyrrolidine-1-carbonyl)piperazine-1-carbonyl]-1,3-thiazol-2-yl}methyl)amine
methyl 2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetate
8-(furan-2-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[1-(5-cyanopyridin-2-yl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
6-(benzyloxy)-4-[(3-fluorophenyl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
5-(1-methylcyclopropanecarbonyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine