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8-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)quinoline
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(propane-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
3-(4-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-2,5-dimethylpyrazine
7,7-dimethyl-2-[1-(2-methylpropyl)-1H-imidazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-4-yl)methanol
4-methyl-7-{[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)amino]methyl}-2H-chromen-2-one
5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}-2-(propylsulfanyl)pyrimidine
5-methyl-4-(1-{1-oxaspiro[4.4]nonan-3-yl}-1H-imidazol-2-yl)-2-(thiophen-2-yl)-1,3-oxazole
2-methyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]thieno[3,2-d]pyrimidin-4-amine
3-[(3-aminoazetidin-1-yl)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
2-[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]-N-benzylacetamide
1-[2-(pyridin-3-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
[(4-{2-[4-(2,2-dimethyloxane-4-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
(2R)-2-amino-1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-phenylethan-1-one
1-[(4aR,8aR)-1-(quinoxaline-6-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
1-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}cyclopentane-1-carboxylic acid
5-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]carbamoyl}amino)-2-methoxy-N-methylbenzamide
6-tert-butyl-N-[2-(dimethylamino)-1-phenylethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(1,3-benzothiazol-2-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidin-4-amine
6-(2,5-dimethylfuran-3-yl)-N-[1-(1H-imidazol-2-yl)ethyl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-propyl-1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2-methoxy-4-methylbenzoyl)piperidine
6-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
3-[3-(morpholin-4-yl)propyl]-1-[4-(1H-pyrazol-4-yl)phenyl]urea
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
4-benzyl-1-[(4-fluoro-3-methylphenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-3-{[(3-methyloxetan-3-yl)methyl]sulfamoyl}-N-(2-methylpropyl)benzamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}cyclopropan-1-amine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yl)ethan-1-one
[1-(5-ethylthiophene-3-carbonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
2-(2-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}phenoxy)acetic acid
2-(4-chlorophenyl)-N-(dimethyl-1,2-oxazol-4-yl)morpholine-4-carboxamide
ethyl 1-[(1-ethylpyrrolidin-2-yl)methyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(4aS,8aR)-6-(5-chlorothiophene-2-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
6-(3-chlorophenyl)-7-(prop-2-en-1-yl)-2-(thiomorpholine-4-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-{methyl[(1-methylpiperidin-2-yl)methyl]amino}pyridine-3-carboxamide
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
1-cyclopropyl-5-oxo-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide
{4-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridin-2-yl}methanol
(3aR,5R,6S,7aS)-2-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
1-{3-[(2-methylphenyl)methoxy]azetidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methoxypyrimidin-2-amine
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(3-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-3-carboxylic acid
(3aR,6aR)-2-[2-(2-chlorophenyl)acetyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3,4-dichlorophenyl)-4-(2-methylpyrimidine-5-carbonyl)morpholine