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(3S,4R)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
1-[1'-(2,5-difluorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(1R,7S)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)propanamide
2-{2-[1-(1,3-benzothiazole-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
6-[3-(methoxymethyl)pyrrolidin-1-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
2-(dimethylamino)-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylphenyl)acetamide
N-(pyridin-2-ylmethyl)-3-{[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
1-(3-fluorophenyl)-6,6-dimethyl-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]oxy}pyrimidine
3-(2-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}ethyl)-2-methyl-1H-indole-5-carbonitrile
N-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
(3E)-1-{2-[5-(azepane-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}pent-3-en-1-one
3-(methylsulfanyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-2-(1-methylpiperidin-2-yl)acetamide
N-[(5-methylpyrazin-2-yl)methyl]-3-[(oxolan-3-yl)sulfamoyl]benzamide
3-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
7-(1,3-benzothiazol-2-yl)-4-[(3-ethyl-1H-pyrazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(dimethylamino)ethyl]-N-ethyl-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[4-(thiophen-2-yl)butanoyl]pyrrolidin-3-yl]acetamide
2-{[3-({2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}carbamoyl)phenyl]amino}acetic acid
1-methyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenylbenzoic acid
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
(2R,6R)-4-[3-(methylsulfanyl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-methyl-1,4-diazepane
3-[(3,4-dimethylpiperazin-1-yl)methyl]-7-methoxy-1,2-dihydroquinolin-2-one
4-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
6-cyclopentyl-N-[(2,4-dimethoxyphenyl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[(diethylamino)methyl]-N-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}pyridine-3-carboxamide
2-(cyclopentylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)morpholine-4-carboxamide
3-(2-chlorophenyl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)pyrrolidine-1-carboxamide
2-[3-(2-methoxyethyl)-5-(2-methyl-5-sulfamoylphenyl)-1H-1,2,4-triazol-1-yl]acetic acid
N,6,8-trimethyl-N-(oxan-2-ylmethyl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-(propan-2-yl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carboxamide
1-(1-benzothiophene-2-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-chloro-5-(1H-pyrazol-1-yl)benzamide
(4-methylpentan-2-yl)[1-(piperidin-3-yl)ethyl]amine
1-[2-methoxy-4-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
(4aR,7aS)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl (2R)-2-({2-[(quinolin-8-yloxy)methyl]-1,3-oxazol-4-yl}formamido)propanoate
6-{octahydropyrrolo[1,2-a]piperazin-2-yl}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-chloro-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-(adamantan-1-yl)-1-(1,4-oxazepan-6-ylmethyl)urea
2-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}-1,4-dihydroquinolin-4-one
5-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridine-5-carbonyl}-1-cyclopentylpiperidin-2-one
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-(1,2-oxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide