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2-(dimethylamino)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(2-methylphenyl)acetamide
2-{[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-5-methyl-1H-1,3-benzodiazole
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(4-propanoylphenoxy)acetamide
(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-propylpiperidin-3-yl)methanol
4-{1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
3-[4-(2-ethyl-2-methyl-3-oxopiperazin-1-yl)-4-oxobutyl]-3,4-dihydroquinazolin-4-one
{1-[({4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)methyl]cyclobutyl}methanol
(4aS,7aR)-1-[2-(naphthalen-1-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenylbutanamide
N-[(2R,3R)-2-hydroxy-1'-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
4-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
2-methyl-1-(4-methyl-1,3-thiazol-2-yl)-4-(2-methylphenyl)piperazine
N-(furan-3-ylmethyl)-N-methyl-3-(1H-pyrazol-1-ylmethyl)benzamide
8-[1-(2-fluorophenyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-2-(1H-imidazol-2-yl)benzamide
N,N-dimethyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]aniline
3-methoxy-2-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
N-[2-(2-fluorophenyl)-1-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methylphthalazine
2-(2-{[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}ethyl)-1,2-dihydrophthalazin-1-one
2-chloro-4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)carbamoyl}amino)-N-(propan-2-yl)benzamide
(4S)-3-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-(propan-2-yl)-1,3-oxazolidin-2-one
1-(2,3-dimethylquinoxalin-6-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
9-(4-hydroxybenzoyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-ethylpiperazin-1-yl)-N-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine
2-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-1,2-oxazinane
1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
2-methyl-4-{5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]furan-2-yl}but-3-yn-2-ol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
1-{1'-[4-(methylamino)pyrimidin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(3-fluorophenyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-amine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
2-ethyl-5-{[4-(1-methylpiperidin-4-yl)piperazin-1-yl]methyl}pyrimidine
5-(2,6-dimethoxyphenyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
1-ethyl-5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-3-(propan-2-yl)-1H-pyrazole
1-{2-oxo-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(azocan-1-yl)-3-[2-methoxy-4-({[(3-methyloxetan-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
methyl 6-oxo-4-(6-phenoxypyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,8-naphthyridine-2-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
3-{[4-(3-aminopentan-3-yl)-1H-1,2,3-triazol-1-yl]methyl}-N,N-dimethylpiperidine-1-sulfonamide
N-({5-[2-methyl-2-(pyrrolidin-1-ylmethyl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-(dimethylamino)-2-(3-methylphenyl)-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)acetamide
2-(adamantan-1-yl)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrimidin-4-ol
N-{1-[1-(2-chlorophenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]propan-2-yl}acetamide
N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,6-dimethyl-4-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl acetate