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2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(2,5-dihydro-1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
4-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
4-chloro-3-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)carbamoyl]amino}-N-methylbenzamide
1-[5-(furan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
N,N-dimethyl-6-{3-[1-(1,3-thiazol-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidin-4-amine
4-methyl-9-(3-phenoxypropanoyl)-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-{4-[5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenyl}acetamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]propan-1-one
4-(2-aminopyridine-4-carbonyl)-1-cyclohexylpiperazin-2-one
2-[3-(dimethylamino)propyl]-9-(2-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-({4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}methyl)benzoate
5-{[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methyl-1H-imidazole
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
N,N-diethyl-1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
5-(5-phenyl-1,2-oxazol-3-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
N,2,6-trimethyl-4-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N3-[(3-fluorophenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-(2-{2-[2-(5-methylfuran-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethylamino)-2-(2-fluorophenyl)-N-[(4-hydroxyphenyl)methyl]acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-methylpyrimidin-2-amine
(4R)-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-3-methyl-1,3-thiazolidine
(furan-2-ylmethyl)(prop-2-en-1-yl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
8-[6-(1-hydroxyethyl)pyridin-2-yl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(4-cyclopentyl-1,4-diazepan-1-yl)-4-(1H-imidazol-1-yl)butan-1-one
N-methyl-N-{2-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}methanesulfonamide
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-6-ethoxyphenol
5-[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)-1,3-thiazole-4-carboxamide
3-(4-fluorophenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(4-methylphenyl)-1H-pyrazole
methyl 4-[4-(6-cyclopropylpyrimidin-4-yl)piperazin-1-yl]benzoate
3-(1-benzyl-1H-imidazol-2-yl)-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
3-cyclopropyl-1-methyl-4-(3-methyl-1-benzothiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
5-(2,6-dimethoxyphenyl)-N-[3-(1H-indol-1-yl)propyl]-1,2,4-triazin-3-amine
N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-3-(1H-pyrazol-1-yl)propanamide
1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-({3-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}methyl)-1H-pyrazole
6-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole
(1S,9aR)-1-{2-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-octahydro-1H-quinolizine
5-{[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}-2,1,3-benzoxadiazole
8-[(2-aminopyridin-3-yl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)-1,3-benzothiazole
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]thiophene-2-sulfonamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-fluoro-4-methylbenzamide
4-cyclopropyl-6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidine
1-(6-cyclopropylpyrimidin-4-yl)-N,N-dimethylazepan-4-amine