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N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-oxopiperidine-3-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-6-(3-fluoro-4-methylbenzenesulfonyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-amino-8-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[(2-methoxyphenyl)methyl]-N3-methyl-N5-(3-methylbutyl)-4-oxo-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(propan-2-yl)-2-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
(1-{5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)methanol
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-3-({1-[(4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-methylbenzamide
1-methyl-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H,2H,3H-imidazo[4,5-c]pyridin-2-one
dimethyl[(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-oxazepan-6-yl)methyl]amine
1-[4-(difluoromethoxy)benzoyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
methyl (2S,4S)-1-methyl-4-(4-phenoxybenzamido)pyrrolidine-2-carboxylate
5-methyl-4-[4-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-2-amine
2-benzyl-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-N-methylpyridine-4-carboxamide
2-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-8-fluoro-1,4-dihydroquinolin-4-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(propan-2-yl)pyrrolidin-3-yl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
4-{[methyl(oxan-4-ylmethyl)amino]methyl}-1H-pyrazole-3-carboxylic acid
1-[(5-chlorothiophen-2-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N-methyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyridin-2-amine
5-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
5-[(isoquinolin-5-yloxy)methyl]-N-(2-methoxybutyl)-1,2-oxazole-3-carboxamide
methyl 4-methoxy-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)benzoate
1-methyl-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[(2,6-difluoro-3-methylphenyl)methyl]-1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
6-methyl-5-{5-[(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)methyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
5-methoxy-N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-indole-2-carboxamide
(3S,9aR)-8-(3-chlorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 4-[(4-chlorophenyl)methyl]-1-[(4-methylphenyl)carbamoyl]piperidine-4-carboxylate
2-(1-benzothiophen-7-yl)-2-(4-ethylpiperazin-1-yl)acetic acid
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-3-propanamidobenzamide
N-(1-hydroxybutan-2-yl)-1-methyl-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)[(2-ethylpyrimidin-4-yl)methyl]methylamine
N-(1-benzyl-1H-pyrazol-3-yl)-2-(4-methyl-1H-indol-1-yl)acetamide
3-(3-{[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrazine-2-carbonitrile
4-(4-chloro-2-hydroxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
(3R,4S)-4-cyclopropyl-1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]pyrrolidin-3-amine
3-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(3-methylbutyl)-6-(1-methylpiperidin-3-yl)-3,4-dihydropyrimidin-4-one
(3-{[1-(3,5-difluoropyridine-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
(2R,3R)-1'-[(3-fluorophenyl)methyl]-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(1H-imidazol-1-yl)-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
2-hydroxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
(3aS,7aR)-5-methyl-2-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide