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(2S,4S)-1-benzyl-4-{[(4-methoxy-3-methylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
8-methyl-5-[4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]quinoline
benzyl({[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
4-(4-{[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
2-{1-[5-(3-methoxyphenyl)furan-2-carbonyl]azetidin-3-yl}pyridine
1-[(4-chlorophenyl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
4-methyl-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1,2,3-thiadiazole-5-carboxamide
8-[(1-ethyl-1H-indol-5-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(methylsulfanyl)-N-(pyridin-3-ylmethyl)propanamide
1-{3-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
methyl 1-[(3R,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
4-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperazine-1-carbonyl}morpholine
N-{[3-methyl-7-(5-phenoxyfuran-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,7-dimethyl-11-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3,7,11-triazaspiro[5.6]dodecane
1-[5-(methoxymethyl)furan-2-carbonyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
2-ethyl-4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)pyrimidine
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
8-[4-(2-hydroxyethyl)piperazine-1-carbonyl]-2-methyl-1,4-dihydroquinolin-4-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
5-[(4-ethoxypiperidin-1-yl)methyl]-2-(4-methoxyphenyl)pyrimidine
3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indazole
3,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
8-methyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(3,4-dimethoxyphenyl)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N,N-dimethyl-5-{1-[(4-methylpyridin-2-yl)methyl]-1H-imidazol-2-yl}pyridin-2-amine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-(9H-fluoren-2-ylmethyl)-4-methyl-1,4-diazepan-5-one
2-(2,3-dimethoxy-5-methylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
4-methyl-N-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-3-(2-methylphenyl)propan-1-one
2-[4-(2-methoxypyridine-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
(1R,3S)-7-[1-(2-fluorophenyl)cyclopropanecarbonyl]-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(4-methoxyphenoxymethyl)-1,3-oxazole
5-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1,2-dimethyl-1H-imidazole
2-{[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-5-methylpyrazine
(3R,4R)-1-(5-ethyl-1,3-oxazole-4-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-{4-[3-(2-methoxyphenyl)propanoyl]-5-methyl-2-oxopiperazin-1-yl}benzonitrile
1-(1-aminocyclobutanecarbonyl)-4-(4-fluoro-2-methylphenoxy)piperidine-4-carboxylic acid
2-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}-1H-1,3-benzodiazole
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
3-(methanesulfonylmethyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidine
N-[(3-hydroxypyrrolidin-3-yl)methyl]-2-[2-(3-methoxyphenyl)ethyl]benzamide
3-{1-[3-(morpholin-4-yl)benzoyl]piperidin-3-yl}benzoic acid
4-(1-ethyl-1H-pyrazol-4-yl)-1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,2,3,6-tetrahydropyridine
3-amino-1-(1H-indol-5-ylmethyl)pyrrolidine-3-carboxylic acid