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4-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4H-chromene-2-carboxamide
(4aS,8aR)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
7-(3-chlorophenyl)-4-(1-ethyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-1,3-diazinane-2,4-dione
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
3-benzyl-4-(3,4-difluorobenzoyl)piperazin-2-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-methoxypyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
[(4-ethynylphenyl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
5-ethyl-N,2-dimethyl-N-[2-(pyridin-2-yl)ethyl]pyrimidin-4-amine
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(4-methoxybenzoyl)-4-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperazine
3-{[1-(3-methoxyphenyl)propan-2-yl]amino}-1-(4-methylpiperidin-1-yl)propan-1-one
1-(3-fluoro-2-hydroxybenzoyl)-3-methylpiperidine-3-carbonitrile
N-(2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)benzamide
4-{[(2,5-difluorophenyl)methyl](1-methoxypropan-2-yl)carbamoyl}benzoic acid
4-methyl-2-{2-oxo-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
1-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)urea
1-[4-(1H-imidazol-1-yl)butanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-(2-methanesulfonamidoethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(2-methyl-1H-imidazol-1-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butanamide
6-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
2-{4-[(2-ethylpyrimidin-4-yl)methyl]piperazin-1-yl}-4-methyl-6-(trifluoromethyl)pyrimidine
4-chloro-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-1H-indole-2-carboxamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[4-({[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}methyl)phenoxy]ethan-1-ol
(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
6-(4-acetylphenyl)-5-cyano-2-methylpyridine-3-carboxylic acid
1-[(2R,3R)-2-hydroxy-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-methylbut-2-en-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(1,2-oxazol-3-ylmethyl)amino]pyridine-3-carboxamide
4-(1,4-dioxan-2-ylmethyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
({4-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
N-butyl-7-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(3-methylfuran-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(2S,4S)-N-ethyl-4-[2-(3-hydroxyphenyl)acetamido]-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}phenol
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-(prop-2-en-1-yl)-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidine-3-carboxylic acid
2-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
2-[1-(3,4-difluorophenyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]morpholine
3-(2-fluorophenyl)-5-(oxolane-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(4-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl)-2-methoxyethan-1-one
1-methyl-8-(propan-2-yl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
1-(2-methylpropyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-amine