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2-[1-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1H-imidazol-2-yl]benzoic acid
2-(1-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
6-methyl-2-({2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
1-{2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-(5-methyl-1,2-oxazol-3-yl)-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}propan-1-one
6-{3-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-cycloheptylethan-1-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-methoxy-N,N-bis(propan-2-yl)-6-(pyrimidin-2-yl)benzamide
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-6-methylphenol
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrimidin-2-yl)-1,4-diazepane
3-(4-methoxy-2-methylphenyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
2-[4-({[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]carbamoyl}amino)piperidin-1-yl]acetamide
3-ethyl-8-[(2,3,4-trimethoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-5-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-indole
1,3-dimethyl-6-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}pyridine
6-(2,6-dimethoxy-4-methylphenyl)-N,N-dimethylpyridazin-3-amine
[(4-fluorophenyl)methyl](oxolan-2-ylmethyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
4-hydroxy-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methyl-4-phenylpiperazine
1-(3,5-dimethyl-4-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]propanamide
2-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
9-[4-(1H-imidazol-1-yl)butanoyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[(2-methyl-2H-1,2,3-benzotriazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
3-(furan-2-yl)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]propanamide
2-cyclopropyl-9-[(5-methyl-1H-imidazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
8-({4-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1,3-oxazol-2-yl}methoxy)quinoline
3-{5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-(2,3-dihydro-1H-inden-2-yl)-2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methylacetamide
[(3R,4R)-1-(4-phenylbenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
6-cyano-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](pyridin-4-ylmethyl)amine
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-(furan-2-ylmethyl)piperidin-4-amine
N,4-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-thiazole-5-carboxamide
4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}thiomorpholine
1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propan-1-one
1-{5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-amido}cyclopentane-1-carboxylic acid
5-[5-(2,4-difluorophenoxymethyl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
2-(2-methoxyphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
N-(2-methyl-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)furan-2-carboxamide
1-(2-{[(3-hydroxypyrrolidin-3-yl)methyl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-{1-[4-(1H-imidazol-1-yl)benzoyl]azetidin-3-yl}pyridine
methyl 5-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate