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N-ethyl-3,4,7-trimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-indole-2-carboxamide
N-cyclopropyl-4-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]sulfamoyl}benzamide
N-(1,3-benzothiazol-2-ylmethyl)-1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,4,6-trimethyl-2-oxo-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-3-phenylpropan-1-ol
(2S)-1-{[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl}pyrrolidine-2-carboxamide
1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidine-3-carbonitrile
methyl (1R,3S,3aR,6aS)-1-[(4-hydroxyphenyl)methyl]-5-methyl-3-(5-methylfuran-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(4aS,8aR)-1-(3-methylbutyl)-6-[3-(1H-pyrrol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-4-methyl-1,3-oxazole
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[4-(ethylamino)pyrimidin-2-yl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(3-hydroxypropyl)-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
4-{[(3R,4S)-3-(2H-1,3-benzodioxol-5-yl)-4-carboxypyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[4-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
2-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]ethan-1-ol
(3R,4S)-4-cyclopropyl-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]pyrrolidin-3-amine
N-{1-[1-benzyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]-2-methylpropyl}acetamide
2-{[(2-methylphenyl)methyl]({[(1s,4s)-4-aminocyclohexyl]methyl})amino}ethan-1-ol
1,2-dimethyl-4-{1-[3-(2-methylphenyl)phenyl]piperidin-4-yl}piperazine
3-hydroxy-3-phenyl-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]pyrrolidine-1-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
3-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(propan-2-yl)piperidine
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-5-methyl-1,2-oxazole
(2S,4S)-N-methyl-4-(4-{[methyl(phenylcarbamoyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,4-diazepan-2-one
(3R)-1-(4-chloro-2-fluorobenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
2-(1H-imidazol-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
4-(4-hydroxypiperidine-1-carbonyl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
(1R,5R)-3-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-3-azabicyclo[3.3.1]nonane
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-imidazole-4-carboxylic acid
N-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-{3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}-1,2,3-thiadiazole
5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-4-yl)propan-2-yl]quinoline-4-carboxamide
3-{[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}benzonitrile
2-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(piperidin-1-ylmethyl)benzamide
1-methyl-5-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-(oxolan-2-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}thiophene-2-carboxamide
1-methyl-4-({5-[(E)-2-phenylethenyl]-1,2,4-oxadiazol-3-yl}methyl)piperazine