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3-[(2-fluorophenyl)formamido]-N-methyl-N-(1H-pyrazol-5-ylmethyl)propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)benzamide
N3-(1-benzylpyrrolidin-3-yl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-{5-[(carbamoylamino)methyl]-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-3-yl}benzamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4,6-dimethylpyrimidin-2-amine
N-{4-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}-2-methoxyacetamide
7-(oxan-4-yl)-2-(pyrimidin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
6-[({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-2-carbonitrile
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
2-(4-methylphthalazin-1-yl)benzamide
1-methyl-4-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
6-[methyl(pyridin-2-ylmethyl)amino]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,N-dimethyl-5-{1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-(3,5-dimethylphenyl)-4-(piperidin-4-yl)piperazin-2-one
[(3R,4R)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
7-[(4-fluorophenyl)methyl]-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
9-[(4-fluoro-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(3,4-dichlorophenyl)piperazine
4-{2-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]propyl}morpholine
N-cyclohexyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(prop-2-yn-1-yl)benzamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(1H-indol-3-yl)ethan-1-one
6-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)-9H-purine
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-(oxolane-2-carbonyl)-1,4-diazepane-1-carboxamide
N-(2-methoxyethyl)-4-methyl-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-[4-(pyridin-4-ylmethyl)piperazin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
4-(2-phenylethyl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylic acid
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-(1-methylpiperidin-4-yl)ethan-1-one
4-(1-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}propan-2-yl)morpholine
5-[(2-chlorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-methylimidazo[1,2-a]pyridine-6-carboxamide
N-[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]-3-[(2-methanesulfonylethyl)sulfamoyl]benzamide
2-(2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethyl)-3,4-dihydroquinazolin-4-one
1-cyclopropanecarbonyl-4-{4-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidine
9-[(3-ethoxyphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
{4-[(2-chlorophenyl)methyl]-1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl}methanol
(4aS,8aR)-1-(3-hydroxypropyl)-6-[3-(pyridin-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(4aS,7aR)-1-(3-fluorobenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-5-({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(1S,5R)-N-[(3-fluorophenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
({5-[1-(1H-indazole-3-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-(1-oxo-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-2-yl)pyrrolidin-2-one
4-(4-methoxy-2-methylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(azepan-1-yl)-2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]ethan-1-one
2-(pyridin-4-yl)-7-(pyrrolidine-1-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-benzyl-N,1-dimethyl-5-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]furan-3-carboxamide
3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
2-{2-[2-(4-fluorophenyl)-1H-imidazol-1-yl]ethyl}-1,3-thiazole
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)urea