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3-{[1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
methyl (2S,4R)-4-(dimethylamino)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)pyrrolidine-2-carboxylate
1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-one
3-[(dimethylamino)methyl]-1-[(5-propylfuran-2-yl)methyl]piperidin-3-ol
1-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
6-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
methyl 2-({[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amino)-4-(methylsulfanyl)butanoate
2-(3-phenylpropyl)-4-(1,2,3-thiadiazole-4-carbonyl)morpholine
2-(2-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}phenyl)-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
5-{[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamido]methyl}thiophene-2-carboxylic acid
N-(2-hydroxyethyl)-N-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-({5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
4-benzyl-1-[5-(methoxymethyl)-1,3,4-oxadiazole-2-carbonyl]piperidin-4-ol
5-{[benzyl(methyl)amino]methyl}-N-[1-(1-methylpiperidin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
4-(4-amino-6,7-dimethoxyquinazolin-2-yl)benzamide
N-(2-{[1-(dimethylcarbamoyl)piperidin-3-yl]formamido}ethyl)pyridine-3-carboxamide
3-(methoxymethyl)-5-({5-[(2E)-pent-2-en-2-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
{1-[(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohexylmethyl)-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
(2S)-N-[2-(4-methoxyphenyl)phenyl]-1-(1H-pyrrole-2-carbonyl)pyrrolidine-2-carboxamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
5-{[({3-[2-(4-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}piperazin-1-yl)ethoxy]phenyl}methyl)(methyl)amino]methyl}pyrrolidin-2-one
2-amino-4-(3,4-dimethoxyphenyl)-6-(3-fluorophenyl)pyridine-3-carbonitrile
2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-imidazole
N3-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N1,N1-dimethylpiperidine-1,3-dicarboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-3-ylmethyl)acetamide
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-(1,3-benzoxazol-2-ylmethyl)-5-(2-chlorophenyl)furan-2-carboxamide
methyl 2-[(4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}phenyl)formamido]acetate
3-(4-chlorophenyl)-N-methyl-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
4-[1-benzyl-5-(2-methanesulfonylethyl)-1H-1,2,4-triazol-3-yl]pyridine
1-(2,5-dihydro-1H-pyrrol-1-yl)-2-{4-[(8-methoxyquinolin-2-yl)methyl]morpholin-3-yl}ethan-1-one
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,7,8-trimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-methoxy-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanol
1-{4-[(2R,3R)-2-hydroxy-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]piperidin-1-yl}ethan-1-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(piperidin-3-ylmethyl)piperidine-4-carboxylic acid
[(3R,4R)-1-(2,5-difluorobenzoyl)-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
3-(1H-imidazol-2-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
[1-(5-chloropyridine-3-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(4aS,8aR)-1-(3-hydroxypropyl)-6-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
(3S,4S)-1-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
3,5,7-trimethyl-2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-indole
1-(propan-2-yl)-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
1-{[1-cyclohexyl-3-(3-methoxyphenoxymethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
1-(1-cyclohexylpiperidine-3-carbonyl)-4-(oxan-4-yl)piperazine