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(2S)-2-acetamido-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}propanamide
2-methyl-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-(cyclohexylmethyl)-5-[4-(4-hydroxyphenyl)piperazine-1-carbonyl]piperidin-2-one
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)cyclobutanecarboxamide
(2-{4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)urea
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
5-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(pyridin-2-yl)acetamide
4-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-2-(propan-2-yl)pyrimidine
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-phenylpropyl)piperazin-2-yl)ethan-1-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-2-ylmethyl)amine
5-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-3-methylthiophene-2-carboxamide
1-[3-(2-methylphenyl)phenyl]-N-[1-(pyrazin-2-yl)propan-2-yl]piperidin-4-amine
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}ethan-1-one
2-(4-ethoxybenzenesulfonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(5-fluoro-2-methylphenyl)methyl]amine
4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-1-(propan-2-yl)pyrrolidin-2-one
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propane-1,2-dione
3-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-1-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
(2R,3R)-1'-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-3-amine
6-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-9H-purin-2-amine
ethyl 4-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazine-1-carboxylate
2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid
3-methoxy-4-methyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-(5-fluoro-2-methoxyphenyl)-4-(1-hydroxy-3-phenylpropyl)piperidine-1-carboxamide
(3S)-3-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}azepan-2-one
1-[(4aR,8aR)-7-[(2-chloro-5-fluorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
N-butyl-2-ethyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
7-methoxy-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3R,4R)-3-cyclopropyl-1-[5-(3-methoxyphenyl)furan-2-carbonyl]-4-methylpyrrolidin-3-ol
methyl 6-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}pyridine-2-carboxylate
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-phenoxypropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)oxan-4-amine
2-(2-ethyl-1H-imidazol-1-yl)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]acetamide
2-methyl-4-{3-methyl-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}pyridine
4-({4-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)piperazine-1-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
6-methyl-5-{2-oxo-2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(2R)-2-hydroxy-3-methylbutanoyl]-1-(2-phenylphenyl)piperazin-2-one
N-[2-(dimethylamino)ethyl]-2,4-dimethyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-5-carboxamide
2-methyl-N-{[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]methyl}propanamide
3-{2-[(3-fluorophenyl)methoxy]phenyl}pyridin-4-amine
7-fluoro-4-[4-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-fluorophenyl)ethan-1-one
4-methyl-3-(1H-pyrazol-3-yl)-1,2-dihydroquinolin-2-one
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide