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1-(4-methylphenyl)-4-[5-(propan-2-yl)thiophene-3-carbonyl]piperazin-2-one
(1S,5R)-3-(1H-indole-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[2-(2-methylphenoxy)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
1-benzyl-3-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}urea
4-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}pyridine
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(4-fluorophenyl)butan-1-one
(3R,4R)-3-cyclobutyl-4-methyl-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-ol
1-methyl-4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepane
3-[2-(4-fluorophenyl)ethyl]-1-(trimethyl-1H-pyrazole-4-carbonyl)piperidine
1-[4-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)phenyl]imidazolidin-2-one
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1'-(oxolane-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]
5-{1-[6-(propan-2-yl)pyridazin-3-yl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-cyclohexyl-5,6-dimethyl-N-[(2-methylphenyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-4-{[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(piperidin-3-yl)benzamide
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetic acid
(3S,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-3-carboxylic acid
2-(cyclopropylmethyl)-9-[2-(1H-imidazol-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(2S)-1-{4-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-4-methyl-1-oxopentan-2-yl]acetamide
6-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,3-benzothiazole
N-methyl-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}thian-4-amine
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
N,5-dimethyl-1-propyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
1-[(1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}-4-(pyrimidin-5-yl)phenol
3-(1,3-benzothiazol-2-yl)-1-[3-(pyrrolidin-1-yl)piperidin-1-yl]propan-1-one
8-(3-hydroxy-4-methoxybenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
2,2-dimethyl-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]oxane-4-carboxamide
ethyl 4-(3-phenylpropyl)-1-(1,2,3-thiadiazole-4-carbonyl)piperidine-4-carboxylate
(3aR,6aR)-2-methyl-N-[2-(2-methylphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)thiomorpholine
N-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carboxamide
8-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-5-fluoroquinoline
1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)pyrrolidin-3-amine
3-propanamido-N-[1-(1H-pyrazol-1-yl)propan-2-yl]benzamide
2-(2,3-dimethylphenoxy)-1-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(4aS,7aR)-1-[(5-chlorothiophen-2-yl)methyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-{3-[1-(dimethylamino)ethyl]phenyl}phenyl)acetic acid
4-[4-(4-methoxyphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
4-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-(furan-3-ylmethyl)-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazine
2-(2-chloro-4-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenoxy)acetamide
1-(2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepan-5-one
3-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide