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5-(azepane-1-carbonyl)-N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(butan-2-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(3,4-dichlorophenyl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
6-(4-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
1-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)-1H-pyrazole
(3S,5R)-1-[3-(3,4-dimethylphenyl)propanoyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
3-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
6-[3-(3,5-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-9H-purine
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(4-hydroxyphenyl)ethyl]-5-methylpiperidin-2-one
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1-phenyl-1H-1,2,3-triazole-5-carboxamide
4-[(6-methylpyridin-3-yl)oxy]-N-[(1R,2S)-2-phenylcyclopropyl]piperidine-4-carboxamide
3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[3-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1H-1,2,4-triazole
1-[2-(3-phenylpropyl)morpholin-4-yl]-3-(thiophen-2-yl)propan-1-one
3-{[(2H-1,3-benzodioxol-4-ylmethyl)amino]methyl}-N-cyclohexyl-N-methylpyridin-2-amine
N,6-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-4-oxo-4H-pyran-2-carboxamide
3-(prop-2-en-1-yl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidine-3-carboxylic acid
(2R,3R)-3-amino-1'-(2-methyl-6-propylpyrimidin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5-(3-acetylphenoxymethyl)-N-[3-(1H-indol-1-yl)propyl]-1,2-oxazole-3-carboxamide
[1-({1-[5-(ethylsulfanyl)thiophene-2-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
2-{[(2R)-2-amino-2-phenylacetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-methoxy-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}pyridin-4-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2,3-dihydro-1H-isoindol-2-yl)acetamide
(2S,4R)-4-amino-N-methyl-1-(piperidine-1-sulfonyl)pyrrolidine-2-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-oxo-4-phenylbutanamide
[(2,2-dimethyloxan-4-yl)methyl](methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-(2-phenylethyl)-2-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}acetamide
2-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-1-(propan-2-yl)-1H-imidazole
8-fluoro-4-oxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1,4-dihydroquinoline-3-carboxamide
1-(2-methyl-5-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
1-(3,4-dihydro-2H-1-benzopyran-3-yl)-2-(1H-imidazol-2-yl)-1H-imidazole
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-(4-methoxy-2-methylphenyl)benzamide
1-{2-[1-(2-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}azepan-2-one
2-{4-[(2-ethoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,4R)-1-(1-methyl-2-oxo-1,2-dihydroquinoline-4-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
2-({[4-(dimethylamino)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-{4-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperazin-1-yl}-N-ethylacetamide
2-(3-chlorophenyl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-[2-(3-fluorophenyl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
2-(2-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-pyrrol-1-yl)pyrimidine
(2R,3R,6R)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
4-[(4-{[1-(pyridine-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[1-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methyl-2,3-dihydropyridazin-3-one
1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
4-[(8-chloro-4-hydroxyquinolin-2-yl)methyl]piperazine-1-sulfonamide
6-(4-chlorophenyl)-N,N-dimethylpyrazine-2-carboxamide