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(1S,9S)-11-[(4-{[(5-methylfuran-2-yl)methyl]amino}quinazolin-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-{4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
(1S,5R)-6-(2-methoxypyridine-3-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[3-(3-methylphenoxy)azetidin-1-yl]-6-(propan-2-yl)pyrimidin-2-amine
1-[1-(2-phenylethyl)-5-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
2-(4-chlorophenyl)-5-cyclobutanecarbonyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-aminoethyl)-N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-(2-methoxyethyl)-8-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(4-methanesulfonylphenyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-[4-({2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]pyridine-3-carbonitrile
3-hydroxy-1-(3-phenylpropyl)-3-{[(piperidin-4-yl)amino]methyl}piperidin-2-one
(3aR,6aR)-2-cyclopentyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(4-chlorophenyl)-4-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)morpholine
ethyl 6-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}pyridine-3-carboxylate
N-[3-(morpholin-4-yl)propyl]-2-(pyrrolidin-1-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-5-(methoxymethyl)furan-2-carboxamide
N-[(2-aminopyridin-3-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyridin-2-amine
2-(4-methoxyphenoxymethyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
dimethyl(2-{2-[1-(6-methylpyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}thian-4-amine
[5-chloro-7-(1H-indazol-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(diphenylmethyl)piperazine
1-(2-methoxyphenyl)-4-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]pyrrolidin-2-one
3,5-dimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-indole-2-carboxamide
6-{[4-(3-ethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
5-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-3-[1-(6-oxo-1,6-dihydropyridine-2-carbonyl)piperidin-3-yl]propanamide
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropan-1-amine
4-(2-methoxyphenoxy)-1-[(5-methylfuran-2-yl)methyl]piperidine
2-cyclohexyl-5-(2,3-dihydro-1H-inden-2-yl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(1R,5S,6S)-6-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-azabicyclo[3.1.0]hexane
4-(pyrimidin-2-yl)-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
2-butyl-8-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(6-methylpyridin-2-yl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
6-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,4-oxazepan-6-ol
(4aS,8aR)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{[2-(2-fluorophenyl)ethyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1R,5R)-3-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
4-(2-methyl-1,3-thiazole-4-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
ethyl 1-{3-[4-(methylsulfanyl)phenyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl}piperidine-3-carboxylate
1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazine
2-(2-{1-[(3E)-4-methylhex-3-en-1-yl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
5-[(2-methylphenyl)methyl]-5-(piperidin-4-yl)-3-(pyrazin-2-ylmethyl)imidazolidine-2,4-dione
2-[1-(cyclohexylmethyl)-4-[4-(trifluoromethyl)pyridin-2-yl]piperazin-2-yl]ethan-1-ol
3-{benzyl[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]amino}-2-methylpropan-1-ol