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5-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-4-methyl-5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-methanesulfonyl-N-[3-(2-phenylacetamido)phenyl]acetamide
3-(4-hydroxyphenyl)-N-methyl-N-(1-methylpyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-6-methyl-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-{2-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2-{2-[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
7-[3-cyclopentyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
2-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)quinolin-8-ol
1-phenyl-1-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
(2R,3R,6R)-5-[(3-fluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2E)-N-{[5-fluoro-7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
2-ethyl-1-(2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-1H-imidazole
[1-(ethylsulfanyl)propan-2-yl]({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
N6-benzyl-N5-(2-methoxyethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
(2-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)urea
1-{3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
2-{[2-(1H-imidazol-4-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-hydroxy-N,2-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
{[4-(1H-pyrazol-1-yl)phenyl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
2-[(3-methoxyphenyl)methyl]-8-(4-methyl-1H-imidazole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
{2-[({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(2-methylphenyl)methyl]amino]ethyl}dimethylamine
1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-(2-methoxyethyl)piperidine
N-methyl-5-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
4-{[3-(1H-1,3-benzodiazol-2-yl)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-4-carboxamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
1-(5-phenyl-1,2-oxazole-3-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
4-benzyl-1-{furo[3,2-c]pyridin-4-yl}piperidine-4-carboxylic acid
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(1S,9aR)-1-{[4-(1H-1,2,3-benzotriazol-1-yl)piperidin-1-yl]methyl}-octahydro-1H-quinolizine
1-(furan-2-carbonyl)-4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-phenylbutanamide
1-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(oxan-4-ylmethyl)amine
(1s,4s)-4-{[methyl(quinolin-6-ylmethyl)amino]methyl}cyclohexan-1-amine
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
8-(6-methylpyridin-2-yl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-(2,4-dichlorophenoxy)ethan-1-one
N-ethyl-6-methoxy-2-oxo-N-(pyridin-4-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
[1-(5-chloro-2-methylpyrimidine-4-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide