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N-(3-phenylprop-2-yn-1-yl)-N-propyl-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanamide
3-{[(1-ethylpyrrolidin-3-yl)methyl]sulfamoyl}-N-methylbenzamide
1-[(2-chloro-6-fluorophenyl)methyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-(morpholin-4-yl)butanamide
8-[6-(dimethylamino)pyrazin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
3-{5-[(4-fluoro-3-methylphenyl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-[5-(1-methylpiperidin-3-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]benzoic acid
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyridin-4-yl)piperazine
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
4,6-dimethyl-1-{2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-1,2-dihydropyrimidin-2-one
5-phenyl-N-[4-(4-{[3-(propan-2-yloxy)propyl]amino}piperidin-1-yl)phenyl]pentanamide
6-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
(4aS,8aS)-2-(6-cyclopropylpyrimidin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
4-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2,7-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
3-{5-[(6-methylpyridin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[3-methyl-1-(pyridin-3-yl)butyl]-1-propylpiperidin-4-amine
methyl (1S,3S,3aR,6aS)-3-(2-ethyl-4-methyl-1H-imidazol-5-yl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-4-(piperidin-1-ylmethyl)benzamide
5-(6-phenylpyridazin-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-(2-methoxyethyl)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(1R)-1-(3-methoxyphenyl)ethyl]-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-methylpiperidine-3-carboxamide
6-(2-chlorophenyl)-N-(2-methoxy-2-methylpropyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N2-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
4-[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridazine
(2S)-4-methanesulfonyl-2-{[5-(morpholin-4-ylmethyl)furan-3-yl]formamido}butanoic acid
2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
2-[4-(1-phenylpiperidin-4-yl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-ethyl-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[(2,3,4-trifluorophenyl)methyl]-1H-imidazole
N,N,5-trimethyl-2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
1,2-diethyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1H-1,3-benzodiazole
N-[2-(oxolan-2-ylmethoxy)phenyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-(3-fluorophenoxy)-1-(furan-2-carbonyl)piperidine
ethyl(furan-3-ylmethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]quinoxaline-6-carboxamide
methyl[1-(pyridin-2-yl)propan-2-yl](thiophen-3-ylmethyl)amine
3-{5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-({[(5-fluoro-1H-indol-2-yl)methyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-methyl-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-chloro-N-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
7-methyl-3-{[(propan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
3-[(cyclobutylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
2-(4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol