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6-cyclopropyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
N-[2-(3,5-dimethylphenoxy)ethyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-(thiophen-3-ylmethyl)propanamide
2-amino-4-(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
methyl N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]carbamate
4-{2-[2-fluoro-6-(propan-2-yloxy)phenyl]pyridine-4-carbonyl}morpholine
4-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-oxazepane
methyl 3-(cyclobutylmethoxy)-5-{[(3R,4R)-4-hydroxypiperidin-3-yl]carbamoyl}benzoate
1-(4-{[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)amino]methyl}phenyl)imidazolidin-2-one
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-[(5-methylthiophen-2-yl)methyl]benzamide
5-methyl-1-phenyl-4-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-2-one
2-methyl-N-(oxan-2-ylmethyl)-7-(pyrazin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(hydroxymethyl)-3-methyl-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
1-[4-(1-butyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
(1R,5S)-8-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3,8-diazabicyclo[3.2.1]octane
N-{[(5-fluoro-2-methylphenyl)carbamoyl]methyl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
4-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl](methyl)amino}-2-methylbutan-2-ol
2-{[1-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
4-methyl-3-{[(1-methyl-2-oxopyrrolidin-3-yl)carbamoyl]amino}benzamide
2-cyclopentyl-9-{2-[methyl(phenyl)amino]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
4-(methoxymethyl)-6-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
3-cyclopropyl-5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1,2,4-oxadiazole
ethyl 1-{1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}piperidine-4-carboxylate
4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-(carbamoylmethyl)-N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-[3-(propan-2-yloxy)propyl]-3-propyl-1H-pyrazole-5-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]propanamide
(3S)-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidine-3-carboxylic acid
2-(oxolan-2-ylmethyl)-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
7-chloro-4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-2-(1H-pyrazol-4-yl)quinoline
N-cyclohexyl-3-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propanamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
3-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-4-ethylpiperazin-2-one
1-(butane-1-sulfonyl)-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-[({2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}amino)methyl]-6,8-dimethylquinolin-4-ol
(3S,5R)-N3-cyclopentyl-N5-(4-fluorophenyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
1,3-dimethyl-N-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-(3-methanesulfonamidopropanoyl)pyrrolidin-3-yl]benzoic acid
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(2S)-1-hydroxypropan-2-yl]-5-methoxybenzamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
3-{1-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]piperidin-3-yl}propanamide
methyl 4-{[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](4-methoxy-4-methylpentan-2-yl)amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3S,4S)-1-(5-methyl-1,2-oxazole-3-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
6-{[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-N-phenylpyrimidin-2-amine